Journal Articles
2024
Diastereoselective Synthesis of N-Heterocycle Substituted Cyclobutanes via Michael Addition onto Cyclobutenes
Emma G. L. Robert and Jerome Waser
Chem. Eur. J. 2024, 30, e202403986. (10.1002/chem.202403986)
Homologation of Alkenyl Carbonyls via a Cyclopropanation/Light-Mediated Selective C-C Cleavage Strategy
Tin V. T. Nguyen, Duncan K. Brownsey, André Bossonnet, Matthew D. Wodrich and Jerome Waser
Angew. Chem., Int. Ed. 2024, 63, e202417719. (10.1002/anie.202417719) Open Access! Raw data
Forging 1,1′-Bicyclopropenyls by Synergistic Au/Ag Dual-Catalyzed Cyclopropenyl Cross-Coupling
Xiangdong Li and Jerome Waser
J. Am. Chem. Soc. 2024, 146, 29712-29719. (10.1021/jacs.4c10996) Open Access! Raw data
Enamine Synthesis via Regiocontrolled 6-endo-dig and 5-exo-dig Tethered Carboamination of Propargylic Alcohols
Helena Solé-Àvila, Mikus Puriņš, Lucas Eichenberger and Jerome Waser
Angew. Chem. Int. Ed. 2024, 63, e202411383. (10.1002/anie.202411383) Open Access! Raw data
Platinum-Catalyzed Isomerization of Cyclopropenes to 1,3-Dienes
Vladyslav Smyrnov, Antonin Homassel, Leander Choudhury, Jerome Waser
Helv. Chim. Acta 2024, 107, e2024000105. (10.1002/hlca.202400105) Open Access! Raw data
Ficini Reaction with Acrylates for the Stereoselective Synthesis of Aminocyclobutanes
Emma G. L. Robert and Jerome Waser
Chem. Eur. J. 2024, 30, e202401810. (10.1002/chem.202401810) Open Access! Raw data
Reaction-Agnostic Featurization of Bidentate Ligands for Bayesian Ridge Regression of Enantioselectivity
Alexandre A. Schoepfer, Ruben Laplaza, Matthew D. Wodrich, Jerome Waser, and Clemence Corminboeuf
ACS Catal. 2024, 14, 9302-9312. (10.1021/acscatal.4c02452) Open Access! Code, Visualizations, Joined publication with LCMD.
Hypervalent Iodine Amino Acid Building Blocks for Bioorthogonal Peptide Macrocyclization
Xing-Yu Liu, Olha Mykhailenko, Adriana Faraone and Jerome Waser
Angew. Chem. Int. Ed. 2024, 63, e202404747. (10.1002/anie.202404747) Open Access! Raw data
Photocatalytic Decarboxylative Functionalization of Cyclopropenes via Cyclopropenium Cation Intermediates
Vladyslav Smyrnov and Jerome Waser
Angew. Chem. Int. Ed. 2024, 63, e202404265. (10.1002/anie.202404265) Open Access! Raw data
Lewis Acid Catalyzed [4+2] Annulation of Bicyclobutanes with Dienol Ethers for the Synthesis of Bicyclo[4.1.1]octanes
Stefano Nicolai and Jerome Waser
Chem. Sci. 2024, 15, 10823-10829. (10.1039/D4SC02767A) Open Access! Raw data
Accessing elusive σ-type cyclopropenium cation equivalents through redox gold catalysis
Xiangdong Li, Matthew D. Wodrich and Jerome Waser
Nat. Chem. 2024, 16, 901-912. (10.1038/s41557-024-01535-8) Open Access! Raw data
Organic Dye Photocatalyzed Synthesis of Functionalized Lactones and Lactams via a Cyclization–Alkynylation Cascade
Diana Cavalli and Jerome Waser
Org. Lett. 2024, 26, 4235–4239. (10.1021/acs.orglett.4c01078) Open Access! Raw data
SOMOphilic alkyne vs radical-polar crossover approaches: The full story of the azido-alkynylation of alkenes
Julien Borrel and Jerome Waser
Beilstein J. Org. Chem. 2024, 20, 701-713. (10.3762/bjoc.20.64) Open Access!
Benzylic C(sp3)−H Azidation: Copper vs Iron Catalysis
Angel Rentería-Gómez, Rubén O. Torres-Ochoa, Pierre Palamini, Raphaël Simonet-Davin, Qian Wang, Jérôme Waser, Jieping Zhu
Helv. Chim. Acta 2024, 107, e202400004. (10.1002/hlca.202400004) Open Access!
Interrupted Polonovski Strategy for the Synthesis of Functionalized Amino Acids and Peptides
Christine Marty, Emmanuelle M. D. Allouche, and Jerome Waser
Org. Lett. 2024, 26, 456-460. (10.1021/acs.orglett.3c03603) Green Access Raw data
2023
Synthesis of Fluorescent Cyclic Peptides via Gold(I)-Catalyzed Macrocyclization
Xing-Yu Liu, Wei Cai, Nathan Ronceray, Aleksandra Radenovic, Beat Fierz and Jerome Waser
J. Am. Chem. Soc. 2023, 145, 26525-26531. (10.1021/jacs.3c09261) Open Access! Raw data
Photocatalyzed [2σ + 2σ] and [2σ + 2π] Cycloadditions for the Synthesis of Bicyclo[3.1.1]heptanes and 5- or 6-Membered Carbocycles
Tin V. T. Nguyen, André Bossonnet, Matthew D. Wodrich and Jerome Waser
J. Am. Chem. Soc. 2023, 145, 25411-25421. (10.1021/jacs.3c09789) Green Access Raw data
Acyl-Ethynylbenziodoxolone (acyl-EBX): Access to Ketene Dithioarylacetals
Pierre Palamini, Julien Borrel, Maël Djaïd, Morgane Delattre and Jerome Waser
Org. Lett. 2023, 25, 7535-7539. (10.1021/acs.orglett.3c02869) Green Access Raw data
One-pot synthesis of functionalized bis(trifluoromethylated)benziodoxoles from iodine(i) precursors
Tobias M. Milzarek, Nieves P. Ramirez, Xing-Yu Liu and Jerome Waser
Chem. Commun. 2023, 59, 12637-12640. (10.1039/D3CC04525K) Green Access Raw data
Cysteine-Cysteine Cross-Conjugation of both Peptides and Proteins with a Bifunctional Hypervalent Iodine-Electrophilic Reagent
Ilias Koutsopetras, Abhaya Kumar Mishra, Rania Benazza, Oscar Hernandez-Alba, Sarah Cianférani, Guilhem Chaubet, Stefano Nicolai and Jerome Waser
Chem. Eur. J. 2023, 29, e202302689. (10.1002/chem.202302689) Open Access!
Semipinacol Rearrangement of Cyclopropenylcarbinols for the Synthesis of Highly Substituted Cyclopropanes
Vladyslav Smyrnov and Jerome Waser
Org. Lett. 2023, 25, 6999-7003. (10.1021/acs.orglett.3c02543) Green Access Raw data
Iron-Catalyzed Synthesis of α-Azido α-Amino Esters via the Alkylazidation of Alkenes
Pierre Palamini, Emmanuelle M. D. Allouche, and Jerome Waser
Org. Lett. 2023, 25, 6791-6795. (DOI: 10.1021/acs.orglett.3c02153) Open Access! Raw data
Azido-alkynylation of alkenes through radical-polar crossover
Julien Borrel and Jerome Waser
Chem. Sci. 2023, 14, 9452-9460. (DOI: 10.1039/D3SC03309K) Open Access! Raw data
Photochemical [2+2] Cycloaddition of Alkynyl Boronates
Oleksandr S. Liashuk, Oleksandr O. Grygorenko, Yulian M. Volovenko and Jerome Waser
Chem. Eur. J. 2023, 29, e202301650. (DOI: 10.1002/chem.202301650) Open Access! Raw data
Synthesis of Trifluoromethylated Alkenes: Hypervalent Iodine Meets High-Valent Copper
Tobias Michael Milzarek and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202306128. (DOI: 10.1002/anie.202306128) Open Access! Raw data
Peptide-Hypervalent Iodine Reagent Chimeras: Enabling Peptide Functionalization and Macrocyclization
Xing-Yu Liu, Xinjian Ji, Christian Heinis and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202306036. (DOI: 10.1002/anie.202306036) Open Access! Raw data
Copper (I)-BOX Catalyzed Asymmetric 3-Component Reaction for the Synthesis of Trifluoromethylated Propargylic Ethers and Anilines
Nieves P. Ramirez and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202305776. (DOI: 10.1002/anie.202305776) Open Access! Raw data
Synthesis of propargyl silanes from terminal alkynes via a migratory Sonogashira reaction
Mikus Purins, Lucas Eichenberger, and Jerome Waser
Chem. Commun. 2023, 59, 7931-7934. (DOI: 10.1039/D3CC01847D ) Open Access! Raw data
Donor-Acceptor Aminocyclobutane Monoesters: Synthesis and Silylium-Catalyzed (4+2) Annulation with Indoles
Emma G. L. Robert, Vincent Pirenne, Matthew D. Wodrich and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202302420. (DOI: 10.1002/anie.202302420 ) Open Access! Raw data
X-Ray and NMR Structural Data of Ethynylbenziodoxolones (EBXs) Reagents and Their Analogues
Eliott Le Du, Nieves P. Ramirez, Stefano Nicolai, Rosario Scopelliti, Farzaneh Fadaei-Tirani, Matthew D. Wodrich, Durga Prasad Hari and Jerome Waser
Helv. Chim. Acta 2023, e202200175. (DOI: 10.1002/hlca.202200175 ) Open Access!
Review Articles
2024
Merging the Reactivity of (Pseudo)cyclic Hypervalent Iodine Reagents and Carbenes or Carbenoids
Nieves P. Ramirez* and Jerome Waser
Synthesis 2024, in press. (DOI: 10.1055/a-2418-8285 ).
Silylium-Catalyzed Activation of Donor-Acceptor Strained Rings and Annulation with Indoles
Emma G. L. Robert and Jerome Waser
Chimia, 2024,78, 234. (10.2533/chimia.2024.234)
2023
Recent progress in alkynylation with hypervalent iodine reagents
Eliott Le Du and Jerome Waser
Chem. Commun. 2023, 59, 1589-1604. (DOI: 10.1039/D2CC06168F ) Open Access!
Publications prior to 2023
Publications 2020-2022
Publications 2017-2019
Publications 2013-2016
Publications 2009-2012