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2024
Arylative Ring Expansion of 3-Vinylazetidin-3-Ols and 3-Vinyloxetan-3-Ols to Dihydrofurans by Dual Palladium and Acid Catalysis
Angewandte Chemie-International Edition
2024-04-12
Vol. 63 , num. 22, p. e202403484.DOI : 10.1002/anie.202403484
Benzylic C(sp3)-H Azidation: Copper vs Iron Catalysis
Helvetica Chimica Acta
2024-03-04
Vol. 107 , num. 3, p. e202400004.DOI : 10.1002/hlca.202400004
Design and Synthesis of C4‐Symmetric Axially Chiral β‐Aryl Porphyrins and Application for Supporting Ir(III)‐Catalyzed Enantioselective C−H Alkylation
Angewandte Chemie International Edition
2024
Vol. 63 , p. e202316393.DOI : 10.1002/anie.202404329
Editing Tetrasubstituted Carbon: Dual C–O Bond Functionalization of Tertiary Alcohols Enabled by Palladium-Based Dyotropic Rearrangement
Journal of the American Chemical Society
2024
Vol. 146 , num. 16, p. 11061-11066.DOI : 10.1021/jacs.4c02924
Catalytic Enantioselective Synthesis of Inherently Chiral Macrocycles by Dynamic Kinetic Resolution
ACS Catalysis
2024
Vol. 14 , num. 7, p. 5140-5146.DOI : 10.1021/acscatal.4c00598
Chalcogen bonding catalysis
Chemical Society Reviews
2024
Vol. 53 , num. 2, p. 586-605.DOI : 10.1039/D3CS00503H
Palladium‐Based Dyotropic Rearrangement Enables A Triple Functionalization of Gem‐Disubstituted Alkenes: An Unusual Fluorolactonization Reaction
Angewandte Chemie International Edition
2024
Vol. 63 , num. 1, p. e202316393.DOI : 10.1002/anie.202316393
2023
Enantioselective Total Synthesis of (-)-Artatrovirenol A
Journal Of The American Chemical Society
2023-10-24
Vol. 145 , num. 44, p. 24408-24415.DOI : 10.1021/jacs.3c09683
Asymmetric Construction of α,α‐Disubstituted Piperazinones Enabled by Benzilic Amide Rearrangement
Angewandte Chemie International Edition
2023-04-24
Vol. 62 , num. 18.DOI : 10.1002/anie.202217954
Terminal Alkynes as One-Carbon Donors in [5+1] Heteroannulation: Synthesis of Pyridines via Ynimine Intermediates and Application in the Total Synthesis of Anibamine B
Angewandte Chemie-International Edition
2023-04-21
DOI : 10.1002/anie.202303537
Divergent Asymmetric Total Synthesis of (−)‐Voacafricines A and B
Angewandte Chemie International Edition
2023-04-11
Vol. 62 , num. 16, p. e202301517.DOI : 10.1002/anie.202301517
Highly Strained Oxygen‐Doped Chiral Molecular Belts of the Zigzag‐Type with Strong Circularly Polarized Luminescence
Angewandte Chemie International Edition
2023-04-03
Vol. 62 , num. 15, p. e202301782.DOI : 10.1002/anie.202301782
Oxidative rearrangement of 1,1-disubstituted alkenes to ketones
Science
2023-03-30
Vol. 379 , num. 6639, p. 1363-1368.DOI : 10.1126/science.adg3182
Enantioselective Total Synthesis of (+)-Stephadiamine
Journal of the American Chemical Society
2023-02-27
Vol. 145 , num. 9, p. 5001-5006.DOI : 10.1021/jacs.3c00884
Inherently chiral calixarenes by a catalytic enantioselective desymmetrizing cross-dehydrogenative coupling
Chemical Science
2023-01-28
Vol. 14 , num. 4, p. 827-832.DOI : 10.1039/D2SC06234H
Organocatalytic Enantioselective Pictet–Spengler Reaction of α‐Ketoesters: Development and Application to the Total Synthesis of (+)‐Alstratine A
Angewandte Chemie International Edition
2023-01-02
Vol. 62 , num. 1, p. e202213831.DOI : 10.1002/anie.202213831
Synthesis and Applications of Ynimines and Enantioselective Total Synthesis of Artatrovirenol A
Lausanne: EPFL2023
p. 446.DOI : 10.5075/epfl-thesis-10563
Diverting the 5-exo-Trig Oxypalladation to Formally 6-endo-Trig Fluorocycloetherification Product through 1,2-O/Pd(IV) Dyotropic Rearrangement
Journal of the American Chemical Society
2023
Vol. 145 , num. 29, p. 15735-15741.DOI : 10.1021/jacs.3c06158
Asymmetric Synthesis of Enantioenriched Zigzag-Type Molecular Belts by Kinetic Resolution and Subsequent Transformations
Organic Letters
2023
Vol. 25 , num. 21, p. 3936-3940.DOI : 10.1021/acs.orglett.3c01314
Dual Photoredox and Copper Catalysis: Enantioselective 1,2-Amidocyanation of 1,3-Dienes
ACS Catalysis
2023
Vol. 13 , num. 11, p. 7523-7528.DOI : 10.1021/acscatal.3c01782
TiCl3-Mediated Reductive Cyclization of Tetrasubstituted Alkenes and Enol Esters Bearing a 2-Nitrophenyl Substituent
Lausanne: EPFL2023
p. 351.DOI : 10.5075/epfl-thesis-10074
Organocatalytic Enantioselective Diels-Alder Reaction of 2-Trifluoroacetamido-1,3-dienes with alpha,beta-Unsaturated Ketones
Angewandte Chemie-International Edition
2023
Vol. 62 , num. 1, p. e202214925.DOI : 10.1002/anie.202214925
2022
Apparent 6-endo-trig Carbofluorination of Alkenes Enabled by Palladium-Based Dyotropic Rearrangement
Angewandte Chemie-International Edition
2022-11-16
Vol. 61 , num. 50, p. e202211470.DOI : 10.1002/anie.202211470
Synthesis of 3-Acyloxyindolenines by TiCl3-Mediated Reductive Cyclization of 2-(ortho-Nitroaryl)-Substituted Enol Esters
Organic Letters
2022-09-19
Vol. 24 , num. 38, p. 7004-7008.DOI : 10.1021/acs.orglett.2c02860
Thiazole Boron Difluoride Dyes with Large Stokes Shift, Solid State Emission and Room-Temperature Phosphorescence
Chemistry-A European Journal
2022-09-19
p. e202202507.DOI : 10.1002/chem.202202507
Migrative Carbofluorination of Saturated Amides Enabled by Pd-Based Dyotropic Rearrangement
Journal of the American Chemical Society
2022-08-02
Vol. 144 , num. 31, p. 14047-14052.DOI : 10.1021/jacs.2c06578
Two-Carbon Ring Expansion of Cyclobutanols to Cyclohexenones Enabled by Indole Radical Cation Intermediate: Development and Application to a Total Synthesis of Uleine
Acs Catalysis
2022-01-05
Vol. 12 , num. 2, p. 1209–1215.DOI : 10.1021/acscatal.1c05621
Catalytic enantioselective Pictet-Spengler reaction of carbonyl compounds: Development and application to the asymmetric total synthesis of indole alkaloids
Lausanne: EPFL2022
p. 331.DOI : 10.5075/epfl-thesis-10066
Taming the radical cation intermediate enabled one-step access to structurally diverse lignans
Nature Communications
2022
Vol. 13 , num. 1, p. 13:3481.DOI : 10.1038/s41467-022-31000-4
Catalytic Enantioselective Pictet–Spengler Reaction of α‐Ketoamides Catalyzed by a Single H‐Bond Donor Organocatalyst
Angewandte Chemie International Edition
2022
Vol. 61 , num. 19, p. e202201788.DOI : 10.1002/anie.202201788
Modular Synthesis of Benzocyclobutenes via Pd(II)-Catalyzed Oxidative [2+2] Annulation of Arylboronic Acids with Alkenes
Journal of the American Chemical Society
2022
Vol. 144 , num. 20, p. 8920–8926.DOI : 10.1021/jacs.2c03565
Asymmetric Total Synthesis of Indole Alkaloids (+)-Condyfoline, (-)-Tubifoline, (+)-Dasycarpidone and (+)-Uleine
Lausanne: EPFL2022
p. 244.DOI : 10.5075/epfl-thesis-9160
2021
Photoredox Catalytic Three-Component Amidoazidation of 1,3-Dienes
Acs Catalysis
2021-09-03
Vol. 11 , num. 17, p. 10871-10877.DOI : 10.1021/acscatal.1c03545
Copper‐Catalyzed Aza‐Sonogashira Cross‐Coupling to Ynimines: Development and Application to the Synthesis of Heterocycles
Angewandte Chemie International Edition
2021-09-01
Vol. 60 , num. 45, p. 24028-24033.DOI : 10.1002/anie.202110901
Enantioselective Total Synthesis of (+)-Nordasycarpidone, (+)-Dasycarpidone, and (+)-Uleine
Helvetica Chimica Acta
2021-07-06
Vol. 104 , num. 8, p. e2100088.DOI : 10.1002/hlca.202100088
C-C bond activation enabled by dyotropic rearrangement of Pd(iv) species
Nature Chemistry
2021-05-24
Vol. 13 , p. 671–676.DOI : 10.1038/s41557-021-00698-y
Visible light photoredox-catalysed remote C-H functionalisation enabled by 1,5-hydrogen atom transfer (1,5-HAT)
Chemical Society Reviews
2021-05-20
Vol. 50 , num. 13, p. 7359-7377.DOI : 10.1039/d0cs00774a
Enantioselective Total Synthesis of (+)-Alstilobanine C, (+)-Undulifoline, and (-)-Alpneumine H
Angewandte Chemie-International Edition
2021-04-23
Vol. 60 , num. 12, p. 12392-12395.DOI : 10.1002/anie.202103580
Selective 1,2-Aminoisothiocyanation of 1,3-Dienes Under Visible-Light Photoredox Catalysis
Angewandte Chemie-International Edition
2021-02-12
Vol. 60 , num. 8, p. 4085-4089.DOI : 10.1002/anie.202014518
Development of remote C-H bond functionalization of redox-active alcohol derivatives and oxidative transformations under photoredox catalysis
Lausanne: EPFL2021
p. 421.DOI : 10.5075/epfl-thesis-9292
Macrocyclization of omega-Isocyanoaldehydes and Towards the Total Synthesis of Jamaicensamide A
Lausanne: EPFL2021
p. 153.DOI : 10.5075/epfl-thesis-8714
Catalytic Enantioselective Synthesis of Morpholinones Enabled by Aza-Benzilic Ester Rearrangement
Journal of the American Chemical Society
2021
Vol. 143 , num. 19, p. 7320-7325.DOI : 10.1021/jacs.1c03915
Iron-Catalysed Remote C(sp3)-H Azidation of O-Acyl Oximes and N -Acyloxy Imidates
CHIMIA International Journal for Chemistry
2021
Vol. 75 , num. 4, p. 329-332.DOI : 10.2533/chimia.2021.329
Natural Product Synthesis Enabled by Domino Processes Incorporating a 1,2-Rearrangement Step
ACS Central Science
2021
Vol. 7 , num. 4, p. 559-569.DOI : 10.1021/acscentsci.1c00075
Catalytic Enantioselective Aminopalladation–Heck Cascade
Angewandte Chemie International Edition
2021
Vol. 60 , num. 13, p. 7093-7097.DOI : 10.1002/anie.202016001
Unified divergent strategy towards the total synthesis of the three sub-classes of hasubanan alkaloids
Nature Communications
2021
Vol. 12 , p. 36.DOI : 10.1038/s41467-020-20274-1
2020
Radical-Cation Cascade to Aryltetralin Cyclic Ether Lignans Under Visible-Light Photoredox Catalysis
Angewandte Chemie-International Edition
2020-09-11
Vol. 59 , num. 47, p. 21195-21202.DOI : 10.1002/anie.202007548
Palladium-Catalyzed Multicomponent Synthesis of Fully Substituted Alkylidene Furanones
Organic Letters
2020-09-04
Vol. 22 , num. 17, p. 7030-7033.DOI : 10.1021/acs.orglett.0c02578
Asymmetric Total Synthesis of (-)-Arborisidine and (-)-19-epi-Arborisidine Enabled by a Catalytic Enantioselective Pictet-Spengler Reaction
Journal Of The American Chemical Society
2020-08-19
Vol. 142 , num. 33, p. 14276-14285.DOI : 10.1021/jacs.0c05804
Synthesis of Benzo[a]carbazoles through Visible Light-Induced Cycloaromatization
Helvetica Chimica Acta
2020-06-29
Vol. 103 , num. 8, p. e2000106.DOI : 10.1002/hlca.202000106
TiCl3-Mediated Synthesis of 2,3,3-Trisubstituted Indolenines: Total Synthesis of (+)-1,2-Dehydroaspidospermidine, (+)-Condyfoline, and (-)-Tubifoline
Angewandte Chemie-International Edition
2020-06-04
Vol. 59 , num. 33, p. 13990-13997.DOI : 10.1002/anie.202005380
Copper-Catalyzed Cyanoalkylative Aziridination of N-Sulfonyl Allylamines
Advanced Synthesis & Catalysis
2020-05-26
Vol. 362 , num. 11, p. 2205-2210.DOI : 10.1002/adsc.202000276
Catalytic Enantioselective Benzilic Ester Rearrangement
Angewandte Chemie-International Edition
2020-04-27
Vol. 59 , num. 18, p. 7261-7265.DOI : 10.1002/anie.202001258
Towards the Sarpagine-Ajmaline-Macroline Family of Indole Alkaloids: Enantioselective Synthesis of an N-Demethyl Alstolactone Diastereomer
Chemistry-A European Journal
2020-03-25
Vol. 26 , num. 21, p. 4866-4873.DOI : 10.1002/chem.202000415
Construction of the Erythrinane Core Skeleton via Asymmetric Catalytic Cascade Reaction of Tertiary Enamides
The Journal of Organic Chemistry
2020
Vol. 85 , num. 20, p. 13211-13219.DOI : 10.1021/acs.joc.0c01992
Copper-Catalyzed 1,2-Methoxy Methoxycarbonylation of Alkenes with Methyl Formate and Synthetic Studies Towards the Total Synthesis of Koumine, Voacafricine A and Voacafricine B
Lausanne: EPFL2020
p. 281.DOI : 10.5075/epfl-thesis-10252
Catalytic Enantioselective Synthesis and Switchable Chiroptical Property of Inherently Chiral Macrocycles
Journal of the American Chemical Society
2020
Vol. 142 , num. 34, p. 14432-14436.DOI : 10.1021/jacs.0c05369
Palladium-Catalyzed Enantioselective Cacchi Reaction: Asymmetric Synthesis of Axially Chiral 2,3-Disubstituted Indoles
Angewandte Chemie International Edition
2020
Vol. 59 , num. 5, p. 2105-2109.DOI : 10.1002/anie.201914049
Functionalization of remote C(sp3)-H bonds enabled by copper-catalyzed coupling of O-acyloximes with terminal alkynes
Nature Communications
2020
Vol. 11 , num. 1, p. 403.DOI : 10.1038/s41467-020-14292-2
Fused N‐Heterocycles with Contiguous Stereogenic Centers Accessed by an Asymmetric Catalytic Cascade Reaction of Tertiary Enamides
Chemistry – A European Journal
2020
Vol. 26 , num. 2, p. 401-405.DOI : 10.1002/chem.201904596
Organocatalytic Double Ugi Reaction with Statistical Amplification of Product Enantiopurity: A Linker Cleavage Approach To Access Highly Enantiopure Ugi Products
Organic Letters
2020
Vol. 22 , num. 2, p. 483-487.DOI : 10.1021/acs.orglett.9b04239
Desymmetrization of Prochiral Cyclopentenes Enabled by Enantioselective Palladium-Catalyzed Oxidative Heck Reaction
Organic Letters
2020
Vol. 22 , num. 1, p. 322-325.DOI : 10.1021/acs.orglett.9b04357
2019
Remote C(sp(3))-H Arylation and Vinylation of N-Alkoxypyridinium Salts to delta-Aryl and delta-Vinyl Alcohols
Chemistry – A European Journal
2019-08-13
Vol. 25 , num. 50, p. 11630-11634.DOI : 10.1002/chem.201902918
Total Synthesis of Alstolactine A & Synthetic Studies Towards Members of Akuammiline Alkaloids
Lausanne: EPFL2019
p. 213.DOI : 10.5075/epfl-thesis-9817
Catalytic Enantioselective Pinacol and Meinwald Rearrangements for the Construction of Quaternary Stereocenters
Journal of the American Chemical Society
2019
Vol. 141 , num. 29, p. 11372-11377.DOI : 10.1021/jacs.9b04551
Copper-Catalyzed 1,2-Methoxy Methoxycarbonylation of Alkenes with Methyl Formate
Angewandte Chemie International Edition
2019
Vol. 58 , num. 30, p. 10305-10309.DOI : 10.1002/anie.201904263
Catalytic Kinetic Resolution by Enantioselective Aromatization: Conversion of Racemic Intermediates of the Barton-Zard Reaction into Enantioenriched 3-Arylpyrroles
Angewandte Chemie International Edition
2019
Vol. 58 , num. 27, p. 9215-9219.DOI : 10.1002/anie.201903589
Iron‐Catalysed Remote C(sp 3 )−H Azidation of O ‐Acyl Oximes and N ‐Acyloxy Imidates Enabled by 1,5‐Hydrogen Atom Transfer of Iminyl and Imidate Radicals: Synthesis of γ‐Azido Ketones and β‐Azido Alcohols
Chemistry – A European Journal
2019
Vol. 25 , num. 40, p. 9477-9484.DOI : 10.1002/chem.201901079
Formal [4+1] Cycloaddition of o ‐Aminobenzyl Chlorides with Isocyanides: Synthesis of 2‐Amino‐3‐Substituted Indoles
Helvetica Chimica Acta
2019
Vol. 102 , num. 3, p. e1900002.DOI : 10.1002/hlca.201900002
Palladium-Catalyzed Synthesis of Ketenimines from Isocyanides and Synthetic Studies Towards the Total Synthesis of Mersilongine
Lausanne: EPFL2019
p. 218.DOI : 10.5075/epfl-thesis-7176
Recent Advances in Catalytic Enantioselective Rearrangement
European Journal of Organic Chemistry
2019
Vol. 2019 , num. 10, p. 1964-1980.DOI : 10.1002/ejoc.201801799
Intramolecular Arylation of Tertiary Enamides through Pd(OAc)2-Catalyzed Dehydrogenative Cross-Coupling Reaction: Construction of Fused N-Heterocyclic Scaffolds and Synthesis of Isoindolobenzazepine Alkaloids
The Journal of Organic Chemistry
2019
Vol. 84 , num. 5, p. 2870-2878.DOI : 10.1021/acs.joc.9b00010
Copper-catalyzed remote C(sp3)–H azidation and oxidative trifluoromethylation of benzohydrazides
Nature Communications
2019
Vol. 10 , num. 1, p. 769.DOI : 10.1038/s41467-019-08741-w
Stereoselective Total Synthesis of Eburnane-Type Alkaloids Enabled by Conformation-Directed Cyclization and Rearrangement
Angewandte Chemie International Edition
2019
Vol. 58 , num. 9, p. 2870-2874.DOI : 10.1002/anie.201813920
Dual Photoredox/Copper Catalysis for the Remote C(sp3 )−H Functionalization of Alcohols and Alkyl Halides by N -Alkoxypyridinium Salts
Angewandte Chemie International Edition
2019
Vol. 58 , num. 7, p. 2139-2143.DOI : 10.1002/anie.201813356
Construction of Quaternary Stereocenters by Palladium-Catalyzed Carbopalladation-Initiated Cascade Reactions
Angewandte Chemie International Edition
2019
Vol. 58 , num. 6, p. 1562-1573.DOI : 10.1002/anie.201806088
Catalytic Atropenantioselective Heteroannulation between Isocyanoacetates and Alkynyl Ketones: Synthesis of Enantioenriched Axially Chiral 3-Arylpyrroles
Angewandte Chemie International Edition
2019
Vol. 58 , num. 5, p. 1494-1498.DOI : 10.1002/anie.201812654
Catalytic Enantioselective α-Ketol Rearrangement
Angewandte Chemie International Edition
2019
Vol. 58 , num. 2, p. 499-503.DOI : 10.1002/anie.201812244
2018
From isonitrile to nitrile via ketenimine intermediate: Palladium-catalyzed 1,1-carbocyanation of ally carbonate by alpha-isocyanoacetate
Tetrahedron
2018-12-06
Vol. 74 , num. 49, p. 6966-6971.DOI : 10.1016/j.tet.2018.10.032
Lewis acid catalyst-steered divergent synthesis of functionalized vicinal amino alcohols and pyrroles from tertiary enamides
Organic Chemistry Frontiers
2018-11-07
Vol. 5 , num. 21, p. 3138-3142.DOI : 10.1039/c8qo00839f
Enantioselective total synthesis of (+)-Peganumine A
Abstracts Of Papers Of The American Chemical Society
2018-08-19
256th National Meeting and Exposition of the American-Chemical-Society (ACS) – Nanoscience, Nanotechnology and Beyond, Boston, MA, Aug 19-23, 2018.Total Synthesis of Alstilobanine C, Undulifoline and Alstilobanine B
Lausanne: EPFL2018
p. 264.DOI : 10.5075/epfl-thesis-8983
Metamorphosis of cycloalkenes for the divergent total synthesis of polycyclic indole alkaloids
Chemical Society Reviews
2018
Vol. 47 , num. 21, p. 7882-7898.DOI : 10.1039/C8CS00454D
Copper-catalyzed methylative difunctionalization of alkenes
Nature Communications
2018
Vol. 9 , num. 1, p. 1995-1999.DOI : 10.1038/s41467-018-06246-6
Chiral phosphoric acid-catalyzed enantioselective three-component Mannich reaction of acyclic ketones, aldehydes and anilines
Tetrahedron
2018
Vol. 74 , num. 38, p. 5143-5149.DOI : 10.1016/j.tet.2018.05.055
Copper-Catalyzed Arylation of Remote C(sp3 )−H Bonds in Carboxamides and Sulfonamides
Angewandte Chemie International Edition
2018
Vol. 57 , num. 40, p. 13288-13292.DOI : 10.1002/anie.201807623
Still Unconquered: Enantioselective Passerini and Ugi Multicomponent Reactions
Accounts of Chemical Research
2018
Vol. 51 , num. 5, p. 1290-1300.DOI : 10.1021/acs.accounts.8b00105
Heteroannulation of Arynes with α-Amino Imides: Synthesis of 2,2-Disubstituted Indolin-3-ones and Application to the Enantioselective Total Synthesis of (+)-Hinckdentine A
Angewandte Chemie International Edition
2018
Vol. 57 , num. 20, p. 5679-5683.DOI : 10.1002/anie.201800746
Indole Alkaloids, Macrocycles and Heterocycles
Lausanne: EPFL2018
p. 627.DOI : 10.5075/epfl-thesis-8477
Copper-Catalyzed Enantioselective Arylative Desymmetrization of Prochiral Cyclopentenes with Diaryliodonium Salts
Angewandte Chemie International Edition
2018
Vol. 57 , num. 10, p. 2721-2725.DOI : 10.1002/anie.201713329
Palladium-Catalyzed Enantioselective Desymmetrizing Aza-Wacker Reaction: Development and Application to the Total Synthesis of (−)-Mesembrane and (+)-Crinane
Angewandte Chemie International Edition
2018
Vol. 57 , num. 7, p. 1995-1909.DOI : 10.1002/anie.201712521
Cooperative Pd/Cu Catalysis: Multicomponent Synthesis of Tetrasubstituted Imidazolones from Methyl α-Isocyanoacetates, Primary Amines, and Aryl(vinyl) Iodides
Organic Letters
2018
Vol. 20 , num. 1, p. 126-129.DOI : 10.1021/acs.orglett.7b03479
2017
“Divergent Total Synthesis of (-)-Rhazinilam, (-)-Leucomidine B and (+)-Leuconodine F” and “Synthetic Studies Towards Sarpagine-Related Indoles”
EPFL2017
p. 249.DOI : 10.5075/epfl-thesis-8156
Catalytic Enantioselective Double Carbopalladation/C−H Functionalization with Statistical Amplification of Product Enantiopurity: A Convertible Linker Approach
Angewandte Chemie International Edition
2017
Vol. 56 , num. 45, p. 14192-14196.DOI : 10.1002/anie.201709133
Copper-Catalyzed Enantioselective Domino Arylation/Semipinacol Rearrangement of Allylic Alcohols with Diaryliodonium Salts
Chemistry – A European Journal
2017
Vol. 23 , num. 53, p. 13037-13041.DOI : 10.1002/chem.201703563
Around isocyanide reactivity
Lausanne: EPFL2017
p. 278.DOI : 10.5075/epfl-thesis-8153
Silver Nitrate-Catalyzed Isocyanide Insertion/Lactamization Sequence to Imidazolones and Quinazolin-4-ones: Development and Application in Natural Product Synthesis
Organic Letters
2017
Vol. 19 , num. 18, p. 4872-4875.DOI : 10.1021/acs.orglett.7b02334
α-Oxo-Ketenimines from Isocyanides and α-Haloketones: Synthesis and Divergent Reactivity
Chemistry – A European Journal
2017
Vol. 23 , num. 52, p. 12744-12748.DOI : 10.1002/chem.201703458
Copper-Catalyzed Three-Component Carboazidation of Alkenes with Acetonitrile and Sodium Azide
Angewandte Chemie International Edition
2017
Vol. 56 , num. 35, p. 10555-10558.DOI : 10.1002/anie.201705353
Palladium-Catalyzed Enantioselective Narasaka-Heck Reaction/Direct C−H Alkylation of Arenes: Iminoarylation of Alkenes
Angewandte Chemie International Edition
2017
Vol. 56 , num. 32, p. 9577-9581.DOI : 10.1002/anie.201705641
Silver-Catalyzed Three-Component 1,1-Aminoacylation of Homopropargylamines: α-Additions for Both Terminal Alkynes and Isocyanides
Angewandte Chemie International Edition
2017
Vol. 56 , num. 27, p. 7958-7962.DOI : 10.1002/anie.201704727
Fluorophores for Excited-State Intramolecular Proton Transfer by an Yttrium Triflate Catalyzed Reaction of Isocyanides with Thiocarboxylic Acids
Angewandte Chemie International Edition
2017
Vol. 56 , num. 23, p. 6599-6603.DOI : 10.1002/anie.201702488
Organocatalytic Enantioselective Acyloin Rearrangement of α-Hydroxy Acetals to α-Alkoxy Ketones
Angewandte Chemie International Edition
2017
Vol. 56 , num. 21, p. 5858-5861.DOI : 10.1002/anie.201701098
Organocatalytic Nucleophilic Addition of Hydrazones to Imines: Synthesis of Enantioenriched Vicinal Diamines
Angewandte Chemie International Edition
2017
Vol. 56 , num. 20, p. 5612-5615.DOI : 10.1002/anie.201702295
Water as a Hydride Source in Palladium-Catalyzed Enantioselective Reductive Heck Reactions
Angewandte Chemie International Edition
2017
Vol. 56 , num. 14, p. 3987-3991.DOI : 10.1002/anie.201700195
To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis
Chemical Society Reviews
2017
Vol. 46 , num. 5, p. 1295-1357.DOI : 10.1039/C6CS00444J
“Palladium-Catalyzed Diamination of Alkynes in Synthesis of Tetracycles” and “Copper-Catalyzed Cyanoalkylation of Unactivated Alkenes”
Lausanne: EPFL2017
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Palladium-Catalyzed Three-Component Reaction of Propargyl Carbonates, Isocyanides, and Alcohols or Water: Switchable Synthesis of Pyrroles and Its Bicyclic Analogues
Organic Letters
2017
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2016
Enantioselective Synthesis of Quaternary α-Amino Acids Enabled by the Versatility of the Phenylselenonyl Group
Chemistry – A European Journal
2016
Vol. 22 , num. 51, p. 18368-18372.DOI : 10.1002/chem.201604781
Organocatalytic Enantioselective Vinylogous Pinacol Rearrangement Enabled by Chiral Ion Pairing
Angewandte Chemie International Edition
2016
Vol. 55 , num. 49, p. 15411-15414.DOI : 10.1002/anie.201609911
Ketenimines from Isocyanides and Allyl Carbonates: Palladium-Catalyzed Synthesis of β,γ-Unsaturated Amides and Tetrazoles
Angewandte Chemie International Edition
2016
Vol. 55 , num. 49, p. 15377-15381.DOI : 10.1002/anie.201609034
Enantioselective Synthesis of (+)-Peganumine A
Journal of the American Chemical Society
2016
Vol. 138 , num. 35, p. 11148-11151.DOI : 10.1021/jacs.6b07846
Copper-catalysed cyanoalkylative cycloetherification of alkenes to 1,3-dihydroisobenzofurans: development and application to the synthesis of citalopram
Chemical Communications
2016
Vol. 52 , num. 74, p. 11100-11103.DOI : 10.1039/C6CC06356J
Synthesis of Diversely Functionalized Oxindoles Enabled by Migratory Insertion of Isocyanide to a Transient σ-Alkylpalladium(II) Complex
Angewandte Chemie International Edition
2016
Vol. 55 , num. 33, p. 9714-9718.DOI : 10.1002/anie.201603950
Copper-Catalyzed Formal [2+2+1] Heteroannulation of Alkenes, Alkylnitriles, and Water: Method Development and Application to a Total Synthesis of (±)-Sacidumlignan D
Angewandte Chemie International Edition
2016
Vol. 55 , num. 32, p. 9249-9252.DOI : 10.1002/anie.201604528
Switchable [3+2] and [4+2] Heteroannulation of Primary Propargylamines with Isonitriles to Imidazoles and 1,6-Dihydropyrimidines: Catalyst Loading Enabled Reaction Divergence
Chemistry – A European Journal
2016
Vol. 22 , num. 24, p. 8332-8338.DOI : 10.1002/chem.201601560
Chiral Phosphoric Acid-Catalyzed Enantioselective Formal [3+2] Cycloaddition of Azomethine Imines with Enecarbamates
Chemistry – A European Journal
2016
Vol. 22 , num. 24, p. 8084-8088.DOI : 10.1002/chem.201601548
Enantioselective Total Synthesis of (−)-Terengganensine A
Angewandte Chemie International Edition
2016
Vol. 55 , num. 22, p. 6556-6560.DOI : 10.1002/anie.201602374
Chiral Phosphoric Acid Catalyzed Asymmetric Ugi Reaction by Dynamic Kinetic Resolution of the Primary Multicomponent Adduct
Angewandte Chemie International Edition
2016
Vol. 55 , num. 17, p. 5282-5285.DOI : 10.1002/anie.201600751
Synthesis of Vinyl Isocyanides and Development of a Convertible Isonitrile
Organic Letters
2016
Vol. 18 , num. 7, p. 1622-1625.DOI : 10.1021/acs.orglett.6b00483
Catalytic Asymmetric Tandem Reaction of Tertiary Enamides: Expeditious Synthesis of Pyrrolo[2,1-a]isoquinoline Alkaloid Derivatives
Angewandte Chemie International Edition
2016
Vol. 55 , num. 11, p. 3799-3803.DOI : 10.1002/anie.201600119
Total Synthesis of (±)-Strictamine
Angewandte Chemie International Edition
2016
Vol. 55 , num. 10, p. 3500-3503.DOI : 10.1002/anie.201511638
Synthesis of Oxazolidin-2-ones by Oxidative Coupling of Isonitriles, Phenyl Vinyl Selenone, and Water
Chemistry – A European Journal
2016
Vol. 22 , num. 7, p. 2278-2281.DOI : 10.1002/chem.201505050
Enantioselective Total Syntheses of (−)-Rhazinilam, (−)-Leucomidine B, and (+)-Leuconodine F
Angewandte Chemie International Edition
2016
Vol. 55 , num. 2, p. 760-763.DOI : 10.1002/anie.201508906
2015
Palladium-Catalyzed Enantioselective Domino Heck/Intermolecular C–H Bond Functionalization: Development and Application to the Synthesis of (+)-Esermethole
Journal of the American Chemical Society
2015
Vol. 137 , num. 51, p. 16028-16031.DOI : 10.1021/jacs.5b11625
An Enantioselective Total Synthesis of (−)-Isoschizogamine
Angewandte Chemie International Edition
2015
Vol. 54 , p. 14937-14940.DOI : 10.1002/anie.201508150
Sulfonamide and Tertiary Amine as Nucleophiles in Pd(II)-Catalyzed Diamination of Alkynes: Synthesis of Tetracyclic Indolobenzothiazine S,S‑Dioxides
Organic Letters
2015
Vol. 17 , num. 21, p. 5256-5259.DOI : 10.1021/acs.orglett.5b02621
Aqueous Titanium Trichloride Promoted Reductive Cyclization of o-Nitrostyrenes to Indoles: Development and Application to the Synthesis of Rizatriptan and Aspidospermidine
Angewandte Chemie International Edition
2015
Vol. 54 , num. 40, p. 11809-11812.DOI : 10.1002/anie.201505713
Synthesis of diverse di- to penta-substituted 1,2-dihydropyridine derivatives from gold(I)-catalyzed intramolecular addition of tertiary enamides to alkynes
Tetrahedron Letters
2015
Vol. 56 , num. 25, p. 3898-3901.DOI : 10.1016/j.tetlet.2015.04.105
Total Synthesis of Aspidosperma Family Indole Alkaloids through the iORC Domino Process
Lausanne: EPFL2015
DOI : 10.5075/epfl-thesis-6607
Total Syntheses of (−)-Mersicarpine, (−)-Scholarisine G, (+)-Melodinine E, (−)-Leuconoxine, (−)-Leuconolam, (−)-Leuconodine A, (+)-Leuconodine F, and (−)-Leuconodine C: Self-Induced Diastereomeric Anisochronism (SIDA) Phenomenon for Scholarisine G and Leuconodines A and C
Journal of the American Chemical Society
2015
Vol. 137 , num. 20, p. 6712-6724.DOI : 10.1021/jacs.5b03619
Synthesis of Functionalized Epoxides by Copper-Catalyzed Alkylative Epoxidation of Allylic Alcohols with Alkyl Nitriles
Organic Letters
2015
Vol. 17 , num. 8, p. 1890-1893.DOI : 10.1021/acs.orglett.5b00571
Pd/C-Catalyzed Cyclizative Cross-Coupling of Two ortho-Alkynylanilines under Aerobic Conditions: Synthesis of 2,3’-Bisindoles
Chemistry – A European Journal
2015
Vol. 21 , num. 20, p. 7413-7416.DOI : 10.1002/chem.201501020
Integrated One-Pot Synthesis of 1,3-Oxazinan-2-ones from Isocyanoacetates and Phenyl Vinyl Selenones
CHIMIA International Journal for Chemistry
2015
Vol. 69 , num. 4, p. 199-202.DOI : 10.2533/chimia.2015.199
Copper-Catalyzed Intermolecular Carboetherification of Unactivated Alkenes by Alkyl Nitriles and Alcohols
Angewandte Chemie International Edition
2015
Vol. 54 , num. 18, p. 5443-5446.DOI : 10.1002/anie.201412357
2-(Methoxycarbonyl)ethyl as a Removable N-Protecting Group: Synthesis of Indoloisoquinolinones by Pd(II)-Catalyzed Intramolecular Diamination of Alkynes
Organic Letters
2015
Vol. 17 , num. 7, p. 1750-1753.DOI : 10.1021/acs.orglett.5b00526
Copper-Catalyzed Cyanomethylation of Allylic Alcohols with Concomitant 1,2-Aryl Migration: Efficient Synthesis of Functionalized Ketones Containing an α-Quaternary Center
Angewandte Chemie International Edition
2015
Vol. 54 , num. 10, p. 3132-3135.DOI : 10.1002/anie.201411657
Enantioselective Synthesis of Putative Lipiarmycin Aglycon Related to Fidaxomicin/Tiacumicin B
Angewandte Chemie International Edition
2015
Vol. 54 , num. 6, p. 1929-1932.DOI : 10.1002/anie.201409475
Multicomponent Reactions in Organic Synthesis
Weinheim, Germany: Wiley-VCH, 2015.ISBN : 978-3-527-33237-3
Tuning the Reactivity of Isocyano Group: Synthesis of Imidazoles and Imidazoliums from Propargylamines and Isonitriles in the Presence of Multiple Catalysts
Angewandte Chemie International Edition
2015
Vol. 54 , num. 4, p. 1293-1297.DOI : 10.1002/anie.201410113
Chiral Calcium–BINOL Phosphate Catalyzed Diastereo- and Enantioselective Synthesis of syn-1,2-Disubstituted 1,2-Diamines: Scope and Mechanistic Studies
Chemistry – A European Journal
2015
Vol. 21 , num. 4, p. 1704-1712.DOI : 10.1002/chem.201405286
Pd-Catalyzed Dehydrogenative Aryl−Aryl Bond Formation via Double C(sp2)−H Bond Activation: Efficient Synthesis of [3,4]-Fused Oxindoles
Organic Letters
2015
Vol. 17 , num. 2, p. 334-337.DOI : 10.1021/ol503442n
2014
Protecting-group-free enantioselective total synthesis of terengganensine A and towards the total synthesis of peganumine A
2014
Advisor(s): J. Zhu
Studies towards the total synthesis of strictamine
2014
Advisor(s): J. Zhu
Thiazoles enabled by discovering new reactivity of isonitriles: synthesis and fluorescence properties
2014
Advisor(s): J. Zhu
On the Formation and Transformation of alpha-Iminonitriles, the Desymmetrization of Bicyclic Bislactones and Total Synthesis of (-)-Leucomidine B and (-)-Rhazinilam
Lausanne: EPFL2014
DOI : 10.5075/epfl-thesis-6489
Plastidic type I signal peptidase 1 is a redox-dependent thylakoidal processing peptidase
Plant Journal
2014
Vol. 80 , num. 4, p. 592-603.DOI : 10.1111/tpj.12655
Isocyanoacetates as Synthetic Platform Towards Natural Products and Biologically Relevant Scaffolds
Lausanne: EPFL2014
DOI : 10.5075/epfl-thesis-6448
“New methods for indoles and [3,4]-fused oxindoles syntheses” and “Copper-catalyzed/mediated difunctionalization of alkenes with alkylnitriles”
Lausanne: EPFL2014
DOI : 10.5075/epfl-thesis-6453
Copper-Mediated/Catalyzed Oxyalkylation of Alkenes with Alkylnitriles
Chemistry – A European Journal
2014
Vol. 20 , num. 45, p. 14633-14636.DOI : 10.1002/chem.201405102
Unified Strategy to Monoterpene Indole Alkaloids: Total Syntheses of (±)-Goniomitine, (±)-1,2-Dehydroaspidospermidine, (±)-Aspidospermidine, (±)-Vincadifformine, and (±)-Kopsihainanine A
Journal of the American Chemical Society
2014
Vol. 136 , num. 42, p. 15102-15108.DOI : 10.1021/ja509329x
Functionalized imidazoliniums from the three-component domino reaction of N-formylmethylcarboxamides with amines and isocyanides
Organic Chemistry Frontiers
2014
Vol. 1 , num. 8, p. 909-913.DOI : 10.1039/C4QO00203B
Mechanistic Study on the Palladium(II)-Catalyzed Synthesis of 2,3-Disubstituted Indoles Under Aerobic Conditions: Anion Effects and the Development of a Low-Catalyst-Loading Process
Chemistry – A European Journal
2014
Vol. 20 , p. 12255-12261.DOI : 10.1002/chem.201403612
Phosphoric Acid Catalyzed Desymmetrization of Bicyclic Bislactones Bearing an All-Carbon Stereogenic Center: Total Syntheses of (−)-Rhazinilam and (−)-Leucomidine B
Angewandte Chemie International Edition
2014
Vol. 53 , num. 37, p. 9926-9930.DOI : 10.1002/anie.201405842
Triple Role of Phenylselenonyl Group Enabled a One-Pot Synthesis of 1,3-Oxazinan-2-ones From α-Isocyanoacetates, Phenyl Vinyl Selenones, and Water
Journal of the American Chemical Society
2014
Vol. 136 , num. 32, p. 11524-11528.DOI : 10.1021/ja506031h
Chiral Phosphoric Acid-Catalyzed Enantioselective Three- Component Aza-Diels-Alder Reactions of Aminopyrroles and Aminopyrazoles
Advanced Synthesis & Catalysis
2014
Vol. 356 , num. 8, p. 1719-1724.DOI : 10.1002/adsc.201400093
From Racemic to Enantioselective Total Synthesis of Trigonoliimines via Development of an Organocatalytic Enantioselective Michael Addition of α-Aryl-α-isocyanoacetate to Vinyl Phenyl Selenone
CHIMIA International Journal for Chemistry
2014
Vol. 68 , num. 4, p. 211-214.DOI : 10.2533/chimia.2014.211
Phosphoric Acid Catalyzed Diastereo- and Enantioselective Synthesis of Substituted 1,3-Diaminotetralins
Organic Letters
2014
Vol. 16 , num. 9, p. 2554-2557.DOI : 10.1021/ol500946w
Copper-catalyzed three-component synthesis of 5-acetamidoimidazoles from carbodiimides, acyl chlorides and isocyanides
Organic Chemistry Frontiers
2014
Vol. 1 , num. 3, p. 240.DOI : 10.1039/c4qo00034j
Three-Component Povarov Reaction–Heteroannulation with Arynes: Synthesis of 5,6-Dihydroindolo[1,2‑a]quinolines
Organic Letters
2014
Vol. 16 , num. 6, p. 1756-1759.DOI : 10.1021/ol500447r
Multicomponent Domino Process: Rational Design and Serendipity
Domino Reactions: Concepts for Efficient Organic Synthesis; Weinheim: Wiley-VCH, 2014. p. 579-610.ISBN : 978-3-527-33432-2
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NIS-Assisted Aza-Friedel-Crafts Reaction with α-Carbamoysulfides as Precursors of
Chemistry – A European Journal
2014
Vol. 20 , num. 13, p. 3621-3625.DOI : 10.1002/chem.201400117
Total Synthesis of (±)-Aspidophylline A
Angewandte Chemie International Edition
2014
Vol. 53 , num. 7, p. 1818-1821.DOI : 10.1002/anie.201310929
2013
Design and Synthesis of 16-Membered Cyclopeptides Active Against Vancomycin-resistant Enterococci (VRE)
CHIMIA International Journal for Chemistry
2013
Vol. 67 , num. 12, p. 916-920.DOI : 10.2533/chimia.2013.916
Enantioselective Total Syntheses of Leuconolam–Leuconoxine–Mersicarpine Group Monoterpene Indole Alkaloids
Journal of the American Chemical Society
2013
Vol. 135 , num. 51, p. 19127-19130.DOI : 10.1021/ja4115192
Iron Chloride-Catalyzed Three-Component Domino Sequences: Syntheses of Functionalized α-Oxy-N-acylhemiaminals and α-Oxyimides
Advanced Synthesis & Catalysis
2013
Vol. 355 , num. 18, p. 3563-3569.DOI : 10.1002/adsc.201300847
Palladium(II)-Catalyzed Cyclizative Cross-Coupling of ortho-Alkynylanilines with ortho-Alkynylbenzamides under Aerobic Conditions
Angewandte Chemie International Edition
2013
Vol. 52 , num. 49, p. 12992-12996.DOI : 10.1002/anie.201307738
Synthesis of Multifunctionalized 1,2,3,4-Tetrahydropyridines, 2,3-Dihydropyridin-4(1H)-ones, and Pyridines from Tandem Reactions Initiated by [5+1] Cycloaddition of N-Formylmethyl-Substituted Enamides to Isocyanides: Mechanistic Insight and Synthetic Application
Chemistry – A European Journal
2013
Vol. 19 , num. 50, p. 16981-16987.DOI : 10.1002/chem.201303221
Catalytic Enantioselective Michael Addition of α-Aryl-α-Isocyanoacetates to Vinyl Selenone: Synthesis of α,α-Disubstituted α-Amino Acids and (+)- and (−)-Trigonoliimine A
Angewandte Chemie International Edition
2013
Vol. 52 , num. 48, p. 12714-12718.DOI : 10.1002/anie.201306663
Palladium-Catalyzed Through-Space C(sp3)-H and C(sp2)-H Bond Activation by 1,4-Palladium Migration: Efficient Synthesis of [3,4]- Fused Oxindoles
Angewandte Chemie International Edition
2013
Vol. 52 , num. 47, p. 12385-12389.DOI : 10.1002/anie.201306532
Heteroannulation of arynes with N-aryl-α-aminoketones for the synthesis of unsymmetrical N-aryl-2,3-disubstituted indoles: an aryne twist of Bischler–Möhlau indole synthesis
Chemical Communications
2013
Vol. 49 , num. 87, p. 10284.DOI : 10.1039/c3cc46361c
Zinc Bromide Promoted Coupling of Isonitriles with Carboxylic Acids To Form 2,4,5-Trisubstituted Oxazoles
Angewandte Chemie International Edition
2013
Vol. 52 , num. 41, p. 10878-10882.DOI : 10.1002/anie.201305506
Tertiary Amines as Synthetic Equivalents of Vinyl Cations: Zinc Bromide Promoted Coupling of Propargylamines with α-Isocyanoacetamides To Give 2,4,5-Trisubstituted Oxazoles Initiated by an Internal Redox Process
Chemistry – A European Journal
2013
Vol. 19 , num. 37, p. 12229-12233.DOI : 10.1002/chem.201302106
Synthetic Study towards Strictamine: The Oxidative Coupling Approach
Synlett
2013
Vol. 24 , p. 1941-1944.DOI : 10.1055/s-0033-1339472
Ugi Four-Component Reaction of Alcohols: Stoichiometric and Catalytic Oxidation/MCR Sequences
Organic Letters
2013
Vol. 15 , num. 11, p. 2854-2857.DOI : 10.1021/ol401181a
Synthesis of Iminonitriles by Oxone/TBAB-Mediated One-Pot Oxidative Three-Component Strecker Reaction
Synthesis
2013
Vol. 45 , num. 10, p. 1380-1386.DOI : 10.1055/s-0032-1316908
Pd(II)-catalyzed intramolecular aminopalladation/direct C–H arylation under aerobic conditions: synthesis of pyrrolo[1,2-a]indoles
Tetrahedron
2013
Vol. 69 , num. 22, p. 4415-4420.DOI : 10.1016/j.tet.2013.01.003
Synthesis of Substituted Pyridines from Cascade [1 + 5] Cycloaddition of Isonitriles to
Journal of the American Chemical Society
2013
Vol. 135 , num. 12, p. 4708-4711.DOI : 10.1021/ja401701x
Palladium-Catalyzed Decarboxylative Vinylation of Potassium Nitrophenyl Acetate: Application to the Total Synthesis of (±)-Goniomitine
Angewandte Chemie International Edition
2013
Vol. 52 , num. 11, p. 3272-3276.DOI : 10.1002/anie.201209970
Synthesis of 3,3-disubstituted oxindoles by one-pot integrated Brønsted base-catalyzed trichloroacetimidation of 3-hydroxyoxindoles and Brønsted acid-catalyzed nucleophilic substitution reaction
Organic & Biomolecular Chemistry
2013
Vol. 11 , num. 9, p. 1533.DOI : 10.1039/c2ob27196f
From natural product to marketed drug: the tiacumicin odyssey
Natural Product Reports
2013
Vol. 30 , num. 1, p. 161.DOI : 10.1039/c2np20080e
2012
Enantioselctive Passerini Reaction
Asymmetric Synthesis – The Essentials II; Weinheim: Wiley-VCH, 2012. p. 95-102.ISBN : 978-3-527-32921-2
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Total Synthesis of Natural Products and the Synergy with Synthetic Methodology
Organic Chemistry-Breakthroughs and Perspectives; Weinheim: Wiley-VCH, 2012. p. 33-79.ISBN : 978-3-527-33377-6
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Copper Catalyzed N-Arylation of Amidines with Aryl Boronic Acids and One-Pot Synthesis of Benzimidazoles by a Chan–Lam–Evans N-Arylation and C–H Activation/C–N Bond Forming Process
Organic Letters
2012
Vol. 14 , num. 23, p. 5980-5983.DOI : 10.1021/ol3028847
Synthesis of Indoles by Copper-Catalyzed Heteroannulation of o-Aminophenylboronic Acid Pinacol Esters with β-Keto Esters
Synthesis
2012
Vol. 44 , num. 24, p. 3811-3814.DOI : 10.1055/s-0032-1316813
Palladium-Catalyzed Coupling of ortho-Alkynylanilines with Terminal Alkynes Under Aerobic Conditions: Efficient Synthesis of 2,3-Disubstituted 3-Alkynylindoles
Angewandte Chemie International Edition
2012
Vol. 51 , num. 49, p. 12311-12315.DOI : 10.1002/anie.201205596
Activation of a C(sp3)H Bond by a Transient s-Alkylpalladium(II) Complex: Synthesis of Spirooxindoles Through a Palladium-Catalyzed Domino Carbopalladation/C(sp3)C(sp3) Bond-Forming Process
Angewandte Chemie International Edition
2012
Vol. 51 , num. 46, p. 11561-11565.DOI : 10.1002/anie.201206267
Amidation of Aldehydes and Alcohols through α-Iminonitriles and a Sequential Oxidative Three-Component Strecker Reaction/Thio-Michael Addition/Alumina-Promoted Hydrolysis Process to Access β-Mercaptoamides from Aldehydes, Amines, and Thiols
Chemistry – A European Journal
2012
Vol. 18 , num. 46, p. 14812-14819.DOI : 10.1002/chem.201202291
Organocatalytic Enantioselective One-Pot Four-Component Ugi-Type Multicomponent Reaction for the Synthesis of Epoxy-tetrahydropyrrolo[3,4-
Chemistry – A European Journal
2012
Vol. 18 , num. 40, p. 12624-12627.DOI : 10.1002/chem.201202174
Synthesis of 4-amino-1,2,3,4-tetrahydropyridine derivatives by intramolecular nucleophilic addition of tertiary enamides to in-situ generated imines
Tetrahedron
2012
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Spirocyclization by Palladium-Catalyzed Domino Heck–Direct C–H Arylation Reactions: Synthesis of Spirodihydroquinolin-2-ones
Organic Letters
2012
Vol. 14 , num. 14, p. 3760-3763.DOI : 10.1021/ol301616w
Development and Application of Isocyanide-based Multicomponent Reactions
Green Synthesis; Weinheim: WIley-VCH, 2012. p. 121-157.ISBN : 978-3-527-32602-0
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Palladium(II)-Catalyzed Intramolecular Diamination of Alkynes under Aerobic Oxidative Conditions: Catalytic Turnover of an Iodide Ion
Angewandte Chemie International Edition
2012
Vol. 51 , num. 21, p. 5170-5174.DOI : 10.1002/anie.201201640
Enantioselective Synthesis of 4-Hydroxytetrahydropyridine Derivatives by Intramolecular Addition of Tertiary Enamides to Aldehydes
Angewandte Chemie International Edition
2012
Vol. 51 , num. 18, p. 4417-4420.DOI : 10.1002/anie.201200459
Synergistic Effect of Palladium and Copper Catalysts: Catalytic Cyclizative Dimerization of ortho-(1-Alkynyl)benzamides Leading to Axially Chiral 1,3-Butadienes
Chemistry – A European Journal
2012
Vol. 18 , num. 19, p. 5864-5868.DOI : 10.1002/chem.201200215
Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Cyclic Enethioureas as Dienophiles: Stereocontrolled Access to Enantioenriched Hexahydropyrroloquinolines
Chemistry – A European Journal
2012
Vol. 18 , num. 19, p. 5869-5873.DOI : 10.1002/chem.201200523
A Concise Total Synthesis of (±)-Trigonoliimine B
Organic Letters
2012
Vol. 14 , num. 5, p. 1338-1341.DOI : 10.1021/ol300249y
Un nouveau venu dans la lutte contre le Clostridium difficile: Les antibiotiques accueillent un nouveau membre
L’Actualité Chimique
2012
num. 360-361, p. 83-89.Exploiting the Divergent Reactivity of Isocyanoacetates: One-Pot Three-Component Synthesis of Functionalized Angular Furoquinolines
European Journal Of Organic Chemistry
2012
p. 475-479.DOI : 10.1002/ejoc.201101567
2011
Unexpected C–C Bond Cleavage: Synthesis of 1,2,4-Oxadiazol-5-ones from Amidoximes with Pentafluorophenyl or Trifluoromethyl Anion Acting as Leaving Group
Organic Letters
2011
Vol. 13 , num. 23, p. 6172-6175.DOI : 10.1021/ol202554m
Trifluoroacetic Acid-Promoted Synthesis of 3-Hydroxy, 3-Amino and Spirooxindoles from α-Keto-N-Anilides
Organic Letters
2011
Vol. 13 , num. 20, p. 5536-5539.DOI : 10.1021/ol202263a
Built-in 5-Aminooxazole as an Internal Activator of the Terminal Carboxylic Acid: An Alternative Access to Macrocyclodepsipeptides
CHIMIA International Journal for Chemistry
2011
Vol. 65 , num. 9, p. 710-714.DOI : 10.2533/chimia.2011.710
Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Enecarbamates as Dienophiles: Highly Diastereo- and Enantioselective Synthesis of Substituted 4-Aminotetrahydroquinolines
Journal of the American Chemical Society
2011
Vol. 133 , num. 37, p. 14804-14813.DOI : 10.1021/ja205891m
A Practical, One-Pot Multicomponent Synthesis of α-Amidosulfides and Their Application as Latent N-Acylimines in the Friedel-Crafts Reaction
European Journal of Organic Chemistry
2011
Vol. 2011 , num. 20-21, p. 3695-3699.DOI : 10.1002/ejoc.201100426
Cinchona Alkaloid-Amides Catalyzed Enantioselective Formal [2+2] Cycloadditions of Allenoates and Imines: Enantioselective Synthesis of 2,4-Substituted Azetidines
Angewandte Chemie -International Edition in English-
2011
Vol. 50 , num. 23, p. 5356-5360.DOI : 10.1002/anie.201100706
Protecting-Group-Free Total Synthesis of (E) and (Z)-Alstoscholarine
Angewandte Chemie -International Edition in English-
2011
Vol. 50 , num. 17, p. 3954-3957.DOI : 10.1002/anie.201100257
Iodo-Carbocyclization of Electron-Deficient Alkenes: Synthesis of Oxindoles and Spirooxindoles
Organic Letters
2011
Vol. 13 , num. 9, p. 2244-2247.DOI : 10.1021/ol2005243
Synthesis of Hydroxylated 3,4-Dihydropyridine-2-ones from Intramolecular Nucleophilic Addition Reaction of Oxirane-containing Tertiary Enamides
Synlett
2011
num. 7, p. 927-930.DOI : 10.1055/s-0030-1259703
Asymmetric Synthesis of 2,4,6-Trideoxy-4-(dimethylamino)-3-C-methyl-Llyxohexopyranose (Lemonose)
Synlett
2011
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Chemistry-A European Journal
2011
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Chiral Calcium Organophosphate-Catalyzed Enantioselective Electrophilic Amination of Enamides
Organic Letters
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2010
Asymmetric Morita–Baylis–Hillman Reaction and Its Aza Analogue
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1-Isocyano-2-nitrobenzene
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1-(2,2-Dimethoxyethyl)-2-isocyanobenzene
e-EROS Encyclopedia of Reagents for Organic Synthesis; 2010.DOI : 10.1002/047084289X.rn01163
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Synthesis of Heterocycles via Multicomponent Reactions II; Berlin: Springer, 2010. p. 1-24.DOI : 10.1007/7081_2010_47
Enantioselective Aza-Morita-Baylis-Hillman Reaction Using Aliphatic alpha -Amidosulfones as Imine Surrogates
Advanced Synthesis & Catalysis
2010
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Copper-promoted N-cyclopropylation of anilines and amines by cyclopropylboronic acid
Chemical Communications
2010
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Zinc Chloride Promoted Formal Oxidative Coupling of Aromatic Aldehydes and Isocyanides to alpha -Ketoamides
Journal of Organic Chemistry
2010
Vol. 75 , num. 8, p. 2748-2751.DOI : 10.1021/jo100302y
Passerini Three-Component Reaction of Alcohols under Catalytic Aerobic Oxidative Conditions
Organic Letters
2010
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Intramolecular Suzuki-Miyaura reaction for the total synthesis of signal peptidase inhibitors, arylomycins A2 and B2
Chemistry–A European Journal
2010
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Palladium-catalyzed domino Heck/cyanation: synthesis of 3-cyanomethyloxindoles and their conversion to spirooxoindoles
Tetrahedron
2010
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Palladium-Catalyzed Carbo-Heterofunctionalization of Alkenes for the Synthesis of Oxindoles and Spirooxindoles
Organic Letters
2010
Vol. 12 , num. 20, p. 4498-4501.DOI : 10.1021/ol101778c
Palladium-Catalyzed Domino Process to Spirooxindoles: Ligand Effect on Aminopalladation versus Carbopalladation
Chemistry–A European Journal
2010
Vol. 16 , num. 20, p. 5863-5867.DOI : 10.1002/chem.201000312
Efficient Synthesis of alpha -Ketoamides via 2-Acyl-5-aminooxazoles by Reacting Acyl Chlorides and alpha -Isocyanoacetamides
Organic Letters
2010
Vol. 12 , num. 4, p. 820-823.DOI : 10.1021/ol902894p
Total synthesis of complestatin (Chloropeptin II)
Angewandte Chemie, International Edition
2010
Vol. 49 , num. 11, p. 2018-2022.DOI : 10.1002/anie.200906797
2009
Invertible Enantioselectivity in 6′-Deoxy-6′-acylamino-beta -isocupreidine-Catalyzed Asymmetric Aza-Morita-Baylis-Hillman Reaction: Key Role of Achiral Additive
Organic Letters
2009
Vol. 11 , num. 20, p. 4648-4651.DOI : 10.1021/ol901920s
Chiral Bronsted Acid-Catalyzed Enantioselective Multicomponent Mannich Reaction: Synthesis of anti-1,3-Diamines Using Enecarbamates as Nucleophiles
Organic Letters
2009
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Synthesis of L-3-hydroxy-4-methoxy-5-methylphenylalanol
Synlett
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IBX/TBAB-mediated oxidation of primary amines to nitriles
Synthesis
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Ugi-post functionalization, from a single set of Ugi-adducts to two distinct heterocycles by microwave-assisted palladium-catalyzed cyclizations: tuning the reaction pathways by ligand switch
Journal of Organic Chemistry
2009
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Synthesis of Pyrroles by Consecutive Multicomponent Reaction/[4 + 1] Cycloaddition of alpha -Iminonitriles with Isocyanides
Organic Letters
2009
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Palladium-catalyzed annulation of acyloximes with arynes (or alkynes): synthesis of phenanthridines and isoquinolines
Angewandte Chemie, International Edition
2009
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Total synthesis of horsfiline: a palladium-catalyzed domino Heck-cyanation strategy
Synlett
2009
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Chiral Bronsted Acid-Catalyzed Enantioselective Three-Component Povarov Reaction
Journal of the American Chemical Society
2009
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Palladium-catalyzed domino N-arylation/carbopalladation/C-H functionalization: three-component synthesis of 3-(diarylmethylene)oxindoles
Tetrahedron Letters
2009
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Combination of lithium chloride and hexafluoroisopropanol for Friedel-Crafts reactions
Synlett
2009
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Asymmetric Total Syntheses of (-)-Renieramycin M and G and (-)-Jorumycin Using Aziridine as a Lynchpin
Organic Letters
2009
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Synthetic Studies on (-)-Lemonomycin: An Efficient Asymmetric Synthesis of Lemonomycinone Amide
Journal of Organic Chemistry
2009
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Catalytic Asymmetric Passerini-Type Reaction: Chiral Aluminum-Organophosphate-Catalyzed Enantioselective alpha -Addition of Isocyanides to Aldehydes
Journal of Organic Chemistry
2009
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Bronsted Acid Catalyzed Enantioselective Three-Component Reaction Involving the alpha Addition of Isocyanides to Imines
Angewandte Chemie, International Edition
2009
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2008
Highly Enantioselective Aza Morita-Baylis-Hillman Reaction Catalyzed by Bifunctional beta -Isocupreidine Derivatives
Journal of the American Chemical Society
2008
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Copper-Mediated N-Cyclopropylation of Azoles, Amides, and Sulfonamides by Cyclopropylboronic Acid
Journal of Organic Chemistry
2008
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Synthesis of dihydrophenanthridines by a sequence of Ugi-4CR and palladium-catalyzed intramolecular C-H functionalization
Beilstein Journal of Organic Chemistry
2008
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Total synthesis of arylomycin A2, a signal peptidase I (SPase I) inhibitor
Synlett
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One-Pot Three-Component Synthesis of alpha -Iminonitriles by IBX/TBAB-Mediated Oxidative Strecker Reaction
Organic Letters
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Synthesis of alpha -keto amides by a molecular-sieves-promoted formal oxidative coupling of aliphatic aldehydes with isocyanides
Angewandte Chemie, International Edition
2008
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Synthesis of diastereomers of complestatin and chloropeptin I: substrate-dependent atropstereoselectivity of the intramolecular Suzuki-Miyaura reaction
Angewandte Chemie, International Edition
2008
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Development of multicomponent and domino reactions based on alpha -isocyanoacetamide and 5-aminooxazole
Seminars in Organic Synthesis, “A. Corbella” Summer School, 33rd, Gargnano, Italy, June 23-27, 2008
2008
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Palladium-Catalyzed Intramolecular C-Arylation of Benzylic Carbon: Synthesis of 3-Benzoxazolylisoindolinones by a Sequence of Ugi-4CR/Postfunctionalization
Journal of Organic Chemistry
2008
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Palladium-Catalyzed Domino Intramolecular N-Arylation/Intermolecular C-C Bond Formation for the Synthesis of Functionalized Benzodiazepinediones
Organic Letters
2008
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Catalytic enantioselective Passerini three-component reaction
Angewandte Chemie, International Edition
2008
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Hafnium Trifluoromethanesulfonate (Hafnium Triflate) as a Highly Efficient Catalyst for Chemoselective Thioacetalization and Transthioacetalization of Carbonyl Compounds
Journal of Organic Chemistry
2008
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Asymmetric Total Synthesis of (-)-Quinocarcin
Journal of the American Chemical Society
2008
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Asymmetric synthesis of 5-(1-hydroxyalkyl)tetrazoles by catalytic enantioselective Passerini-type reactions
Angewandte Chemie, International Edition
2008
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2007
Modulating the reactivity of alpha -isocyanoacetates: multicomponent synthesis of 5-methoxyoxazoles and furopyrrolones
Angewandte Chemie, International Edition
2007
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Rapid synthesis of cyclodepsipeptides containing a sugar amino acid or a sugar amino alcohol by a sequence of a multicomponent reaction and acid-mediated macrocyclization
Journal of Organic Chemistry
2007
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Total synthesis of the marine natural product (-)-cribrostatin 4 (renieramycin H)
Angewandte Chemie, International Edition
2007
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Lithium bromide-promoted three-component synthesis of oxa-bridged tetracyclic tetrahydroisoquinoline derivatives
Heterocycles
2007
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Synthesis of DEFG ring of complestatin and chloropeptin I: highly atropdiastereoselective macrocyclization by intramolecular Suzuki-Miyaura reaction
Organic Letters
2007
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The enantioselective Morita-Baylis-Hillman reaction and its aza counterpart
Angewandte Chemie, International Edition
2007
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IBX-mediated oxidative Ugi-type multicomponent reactions: application to the N and C1 functionalization of tetrahydroisoquinoline
Angewandte Chemie, International Edition
2007
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Palladium-catalyzed three-component synthesis of 3-(diarylmethylene)oxindoles through a domino Sonogashira/carbopalladation/C-H activation/C-C bond-forming sequence
Angewandte Chemie, International Edition
2007
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Palladium-catalyzed enantioselective domino Heck-cyanation sequence: development and application to the total synthesis of esermethole and physostigmine
Chemistry–A European Journal
2007
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Ammonium Chloride Promoted Three-Component Synthesis of 5-Iminooxazoline and Its Subsequent Transformation to Macrocyclodepsipeptide
Organic Letters
2007
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Synthesis of Protected Chiral Vicinal Diaminoalcohols by Diastereoselective Intramolecular Benzylic Substitution from Bistrichloroacetimidates
Organic Letters
2007
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Asymmetric Lewis acid catalyzed addition of isocyanides to aldehydes. Synthesis of 5-amino-2-(1-hydroxyalkyl)oxazoles
European Journal of Organic Chemistry
2007
num. 24, p. 4076-4080.DOI : 10.1002/ejoc.200700340
Chiral Salen-Aluminum Complex as a Catalyst for Enantioselective alpha -Addition of Isocyanides to Aldehydes: Asymmetric Synthesis of 2-(1-Hydroxyalkyl)-5-aminooxazoles
Organic Letters
2007
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New Frontiers in Asymmetric Catalysis edited by Koichi Mikami and Mark Lautens
Angewandte Chemie, International Edition
2007
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Preparation of ecteinascidin alkaloids, such as ecteinascidins 583 and 597
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- US2009171080 (A1)
- JP2009512662 (A)
- EP1937689 (A2)
- WO2007045686 (A3)
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2006
Rapid access to oxindoles by the combined use of an Ugi four-component reaction and a microwave-assisted intramolecular Buchwald-Hartwig amidation reaction
Organic Letters
2006
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5-aminooxazole as an internal traceless activator of C-terminal carboxylic acid: rapid access to diversely functionalized cyclodepsipeptides
Chemistry–A European Journal
2006
Vol. 12 , num. 4, p. 1174-1184.DOI : 10.1002/chem.200500703
Asymmetric total syntheses of ecteinascidin 597 and ecteinascidin 583
Angewandte Chemie, International Edition
2006
Vol. 45 , num. 47, p. 8028-8032.DOI : 10.1002/anie.200603179
Synthetic studies on ecteinascidin 743 (Et 743): asymmetric synthesis of a highly oxygenated tetrahydroisoquinoline via a key phenolic Mannich reaction
Synthesis
2006
num. 23, p. 4081-4086.DOI : 10.1055/s-2006-950343
Total Synthesis of Ecteinascidin 743
Journal of the American Chemical Society
2006
Vol. 128 , num. 1, p. 87-89.DOI : 10.1021/ja0571794
Synthetic studies towards (-)-lemonomycin, synthesis of fused tetracycles
Synlett
2006
num. 11, p. 1691-1694.DOI : 10.1055/s-2006-944225
Aziridinium from N,N-dibenzyl serine methyl ester: Synthesis of enantiomerically pure beta -amino and alpha ,beta -diamino esters
Organic Letters
2006
Vol. 8 , num. 10, p. 2183-2186.DOI : 10.1021/ol060700u
Rapid synthesis of cyclopeptide alkaloid-like para-cyclophanes by combined use of Ugi-4CR and intramolecular SNAr reaction
QSAR & Combinatorial Science
2006
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Mono alkylation of alpha -isocyano acetamide to its higher homologues
Synlett
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Importance of the structure of vancomycin binding pocket in designing compounds active against vancomycin-resistant enterococci (VRE)
Journal of Antibiotics
2006
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Palladium-Catalyzed, Modular Synthesis of Highly Functionalized Indoles and Tryptophans by Direct Annulation of Substituted o-Haloanilines and Aldehydes
Journal of Organic Chemistry
2006
Vol. 71 , num. 20, p. 7826-7834.DOI : 10.1021/jo061471s
Design and synthesis of simple macrocycles active against vancomycin-resistant Enterococci (VRE)
Chemistry–A European Journal
2006
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Synthesis of 4-nitrophenyl sulfones and application in the modified Julia olefination
Synlett
2006
num. 8, p. 1255-1259.DOI : 10.1055/s-2006-939682
Alcohols in isonitrile-based multicomponent reaction: Passerini reaction of alcohols in the presence of o-iodoxybenzoic acid
Angewandte Chemie, International Edition
2006
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Synthesis of 3-(Diarylmethylenyl)oxindole by a Palladium-Catalyzed Domino Carbopalladation/C-H Activation/C-C Bond-Forming Process
Organic Letters
2006
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One-pot synthesis of macrocycles by a tandem three-component reaction and intramolecular [3+2] cycloaddition
Organic Letters
2006
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Preparation of beta-amino or alpha ,beta-diamino esters derived from serine
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2005
Multicomponent Reaction, an overview
Recent progress in Organic Synthesis; Beijing: Chemical Industry Press, 2005.ISBN : 7-5025-7204-X
One or More CH Bond(s) Formed by Substitution: Reduction of C-N, -P, -Arsenic, -Antimony, -Bismuth, -Carbon, -Silicon, -Germanium, -Boron, and –Metal Bonds
Comprehensive Organic Functional Group Transformations II; Cambridge: Elsevier, 2005. p. 31-78.ISBN : 978-0-08-044256-3
Nouveau Composes Chiraux Dérives d’une Diamine ou d’un Aminoalcool, Monosulfonylés et carbonylés Porteurs d’un Groupe Pyrrolidinyle. Leur Préparation et Leurs Applications en Catalyse Asymétrique
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2005
One or more C-H bond(s) formed by substitution: reduction of carbon-nitrogen, -phosphorus, -arsenic, -antimony, -bismuth, -carbon, -boron and -metal bonds
Comprehensive Organic Functional Group Transformations II; Amsterdam: Elsevier Pergamon, 2005. p. 31-78.DOI : 10.1016/B0-08-044655-8/00002-7
Conformation-directed macrocyclization reactions
European Journal of Organic Chemistry
2005
num. 10, p. 1949-1964.DOI : 10.1002/ejoc.200400751
Exploiting the Dual Reactivity of o-Isocyanobenzamide: Three-Component Synthesis of 4-Imino-4H-3,1-benzoxazines
Organic Letters
2005
Vol. 7 , num. 23, p. 5285-5288.DOI : 10.1021/ol052239w
Mild Oxidative One-Carbon Homologation of Aldehyde to Amide
Journal of the American Chemical Society
2005
Vol. 127 , num. 19, p. 6926-6927.DOI : 10.1021/ja0511220
Synthetic Studies toward Ecteinascidin 743
Journal of Organic Chemistry
2005
Vol. 70 , num. 11, p. 4397-4408.DOI : 10.1021/jo050408k
Asymmetric synthesis of protected γ-carboxy-L-glutamic acid
Synlett
2005
num. 5, p. 851-853.DOI : 10.1055/s-2005-863734
Total synthesis of mauritines A, B, C, and F: Cyclopeptide alkaloids with a 14-membered paracyclophane unit
Chemistry–A European Journal
2005
Vol. 11 , num. 9, p. 2668-2679.DOI : 10.1002/chem.200401070
Multicomponent synthesis of epoxy-tetrahydronaphthyridine and structural diversification by subsequent fragmentation
Tetrahedron
2005
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Synthesis of alpha -isocyano-alpha -alkyl(aryl)acetamides and their use in the multicomponent synthesis of 5-aminooxazole, pyrrolo[3,4-b]pyridin-5-one and 4,5,6,7-tetrahydrofuro[2,3-c]pyridine
Synthesis
2005
num. 1, p. 161-165.DOI : 10.1055/s-2004-831225
Three-component synthesis of polysubstituted 6-azaindolines and its tricyclic derivatives
Organic Letters
2005
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Synthesis of ring-A-substituted tryptophan by a palladium-catalyzed heteroannulation reaction
Synlett
2005
num. 16, p. 2469-2472.DOI : 10.1055/s-2005-917079
Identification of synthetic compounds active against VRE: the role of the lipidated aminoglucose and the structure of glycopeptide binding pocket
Bioorganic & Medicinal Chemistry Letters
2005
Vol. 15 , num. 20, p. 4594-4599.DOI : 10.1016/j.bmcl.2005.06.098
Microwave-Assisted Intramolecular Suzuki-Miyaura Reaction to Macrocycle, a Concise Asymmetric Total Synthesis of Biphenomycin B
Organic Letters
2005
Vol. 7 , num. 14, p. 2981-2984.DOI : 10.1021/ol050949w
Synthesis of beta -amino-alpha -hydroxy esters and beta -amino-alpha -azido ester by Sharpless asymmetric aminohydroxylation, byproducts analysis
Journal of Organic Chemistry
2005
Vol. 70 , num. 7, p. 2847-2850.DOI : 10.1021/jo047772o
Design and synthesis of macrocycles active against vancomycin-resistant enterococci (VRE): the interplay between D-Ala-D-Lac binding and hydrophobic effect
Bioorganic & Medicinal Chemistry Letters
2005
Vol. 15 , num. 3, p. 743-746.DOI : 10.1016/j.bmcl.2004.11.014
Synthesis of Chiral Vicinal Diamines by Highly Diastereoselective Three-Component Phenolic Mannich Reaction: Temperature-Dependent Stereodivergency
Organic Letters
2005
Vol. 7 , num. 8, p. 1641-1644.DOI : 10.1021/ol050334z
A three-component synthesis of (1,3-oxazol-2-yl)-1,2-dihydro(iso)quinoline and its further structural diversifications
Synlett
2005
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Multicomponent Reactions
Weinheim: Wiley, 2005.ISBN : 3-527-30806-7
2004
Reeve’s synthesis of 2-imino-4-thiazolidinone from alkyl (aryl) trichloromethylcarbinol revisited, a three-component process from aldehyde, chloroform, and thiourea
Tetrahedron Letters
2004
Vol. 45 , num. 23, p. 4449-4452.DOI : 10.1016/j.tetlet.2004.04.055
Ammonium Chloride Promoted Ugi Four-Component, Five-Center Reaction of alpha -Substituted alpha -Isocyano Acetic Acid: A Strong Solvent Effect
Organic Letters
2004
Vol. 6 , num. 25, p. 4771-4774.DOI : 10.1021/ol0479388
Strained-Cyclophane-Induced beta -Turn Template: Design, Synthesis, and Spectroscopic Characterization
Organic Letters
2004
Vol. 6 , num. 18, p. 3183-3186.DOI : 10.1021/ol0488439
Palladium- and Copper-Catalyzed Synthesis of Medium- and Large-Sized Ring-Fused Dihydroazaphenanthrenes and 1,4-Benzodiazepine-2,5-diones. Control of Reaction Pathway by Metal-Switching
Journal of the American Chemical Society
2004
Vol. 126 , num. 44, p. 14475-14484.DOI : 10.1021/ja047472o
Truncated diastereoselective Passerini reaction, a rapid construction of polysubstituted oxazole and peptides having an alpha -hydroxy-beta -amino acid component
Tetrahedron
2004
Vol. 60 , num. 22, p. 4879-4885.DOI : 10.1016/j.tet.2004.03.084
A short enantioselective synthesis of protected L-3-hydroxy-4-methoxy-5-methyl phenylalanine and its corresponding aldehyde – a common subunit of ecteinascidin-743, safracin and congeners
Synlett
2004
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Synthesis of Polysubstituted 4,5,6,7-Tetrahydrofuro[2,3-c]pyridines by a Novel Multicomponent Reaction
Organic Letters
2004
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A short synthesis of (-)-deoxoprosophylline
Heterocycles
2004
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2003
Total synthesis of an atropdiastereomer of RP-66453 and determination of its absolute configuration
Angewandte Chemie, International Edition
2003
Vol. 42 , num. 35, p. 4238-4241.DOI : 10.1002/anie.200351996
Rapid and diverse route to natural product-like biaryl ether containing macrocycles
Tetrahedron
2003
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Solid-phase synthesis of natural product-like macrocycles by a sequence of Ugi-4CR and SNAr-based cycloetherification
Tetrahedron Letters
2003
Vol. 44 , num. 30, p. 5575-5578.DOI : 10.1016/S0040-4039(03)01378-9
One-pot synthesis of polyheterocycles by a palladium-catalyzed intramolecular N-arylation/C[bond]H activation/aryl[bond]aryl bond-forming domino process
Angewandte Chemie, International Edition
2003
Vol. 42 , num. 39, p. 4774-7.DOI : 10.1002/anie.200351923
Synthetic studies on ecteinascidin 743: rapid access to the fully functionalized tetrahydroisoquinoline with a bridged 10-membered sulfur containing macrocycle
Chemical Communications
2003
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From central to planar chirality, the first example of atropenantioselective cycloetherification
Organic & Biomolecular Chemistry
2003
Vol. 1 , num. 1, p. 30-32.DOI : 10.1039/b208905j
A one-pot four-component (ABC2) synthesis of macrocycles
Angewandte Chemie, International Edition
2003
Vol. 42 , num. 7, p. 811-814.DOI : 10.1002/anie.200390216
Asymmetric synthesis of orthogonally protected (2S,4R)- and (2S,4S)-4-hydroxyornithine
Synlett
2003
num. 10, p. 1455-1458.DOI : 10.1055/s-2003-40840
Allo-aromadendrane- and picrotoxane-type sesquiterpenes from Dendrobium moniliforme
Planta Medica
2003
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Synthesis of isocyano peptides by dehydration of the N-formyl derivatives
Synlett
2003
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Recent developments in the isonitrile-based multicomponent synthesis of heterocycles
European Journal of Organic Chemistry
2003
num. 7, p. 1133-1144.DOI : 10.1002/ejoc.200390167
2002
Studies toward the total synthesis of RP-66453
Tetrahedron Letters
2002
Vol. 43 , num. 14, p. 2577-2580.DOI : 10.1016/S0040-4039(02)00307-6
N-Carbamate-Assisted Stereoselective Synthesis of Chiral Vicinal Amino Sulfides
Organic Letters
2002
Vol. 4 , num. 7, p. 1235-1238.DOI : 10.1021/ol025743z
Synthesis of furoquinolines by a multicomponent domino process
Angewandte Chemie, International Edition
2002
Vol. 41 , num. 19, p. 3633-3635.DOI : 10.1002/1521-3773(20021004)41:19<3633::AID-ANIE3633>3.0.CO;2-T
Rapid access to tetracyclic ring system of lennoxamine type natural product by combined use of a novel three-component reaction and Pummerer cyclization
Chemical Communications
2002
num. 20, p. 2448-2449.DOI : 10.1039/B207179G
Multicomponent domino process to oxa-bridged polyheterocycles and pyrrolopyridines, structural diversity derived from work-up procedure
Tetrahedron
2002
Vol. 58 , num. 32, p. 6351-6358.DOI : 10.1016/S0040-4020(02)00634-8
A five-component synthesis of hexasubstituted benzenes
Angewandte Chemie, International Edition
2002
Vol. 41 , num. 22, p. 4291-4294.DOI : 10.1002/1521-3773(20021115)41:22<4291::AID-ANIE4291>3.0.CO;2-D
Ammonium Chloride-Promoted Four-Component Synthesis of Pyrrolo[3,4-b]pyridin-5-ones
Journal of the American Chemical Society
2002
Vol. 124 , num. 11, p. 2560-2567.DOI : 10.1021/ja017563a
Wilkinson’s Catalyst Catalyzed Selective Hydrogenation of Olefin in the Presence of an Aromatic Nitro Function: A Remarkable Solvent Effect
Journal of Organic Chemistry
2002
Vol. 67 , num. 9, p. 3163-3164.DOI : 10.1021/jo025595q
A Convergent Approach to Cyclopeptide Alkaloids: Total Synthesis of Sanjoinine G1
Journal of the American Chemical Society
2002
Vol. 124 , num. 4, p. 583-590.DOI : 10.1021/ja0170807
2001
An autoxidative approach to 1,2,3,4-tetrahydroisoquinolin-1-one and tetrahydro-β-carbolin-1-one
Tetrahedron Letters
2001
Vol. 42 , num. 20, p. 3427-3430.DOI : 10.1016/S0040-4039(01)00482-8
Asymmetric total synthesis of (-)-deoxoprosophylline
Tetrahedron Letters
2001
Vol. 42 , num. 20, p. 3431-3434.DOI : 10.1016/S0040-4039(01)00483-X
Studies on the Total Synthesis of RP 66453: Synthesis of Fully Functionalized 15-Membered Biaryl-Containing Macrocycle
Organic Letters
2001
Vol. 3 , num. 13, p. 2061-2064.DOI : 10.1021/ol016021v
A Rapid Access to Biaryl Ether Containing Macrocycles by Pairwise Use of Ugi 4CR and Intramolecular SNAr-Based Cycloetherification
Organic Letters
2001
Vol. 3 , num. 25, p. 4079-4082.DOI : 10.1021/ol0168420
Three component synthesis of oxa-bridged tetracyclic tetrahydroquinolines
Chemical Communications
2001
num. 17, p. 1684-1685.DOI : 10.1039/b104317j
4-Nitrophenyltriflate
e-EROS Encyclopedia of Reagents for Organic Synthesis; 2001.DOI : 10.1002/047084289X.rn00477
A Novel Multicomponent Synthesis of Polysubstituted 5-Aminooxazole and Its New Scaffold-Generating Reaction to Pyrrolo[3,4-b]pyridine
Organic Letters
2001
Vol. 3 , num. 6, p. 877-880.DOI : 10.1021/ol007055q
Activation of a terminal carboxylic acid by an internal oxazole: a novel synthesis of macrocyclodepsipeptide
Journal of the American Chemical Society
2001
Vol. 123 , num. 27, p. 6700-6701.DOI : 10.1021/ja015854d
1,3,4,6,7,8-Hexahydro-1-methyl-2H-pyr- imido[1,2-a]pyrimidine (MTBD)
e-EROS Encyclopedia of Reagents for Organic Synthesis; 2001.DOI : 10.1002/047084289X.rn00329.pub2
Polymer-Supported 1,5,7-Triazabicyclo[4.4.0]dec-5-ene (PTBD)
e-EROS Encyclopedia of Reagents for Organic Synthesis; 2001.DOI : 10.1002/047084289X.rn00330
2000
An efficient stereoselective and stereodivergent synthesis of (2R,3R)- and (2R,3S)-3-hydroxypipecolic acids
Tetrahedron Letters
2000
Vol. 41 , num. 36, p. 7033-7036.DOI : 10.1016/S0040-4039(00)01207-7
The first total synthesis of mauritine-A
Tetrahedron Letters
2000
Vol. 41 , num. 40, p. 7645-7649.DOI : 10.1016/S0040-4039(00)01335-6
An efficient total synthesis of K-13, a non-competitive inhibitor of ACE I
Tetrahedron Letters
2000
Vol. 41 , num. 23, p. 4573-4577.DOI : 10.1016/S0040-4039(00)00695-X
Contribution to total synthesis of Vancomycin and Teicoplanin
L’Actualité Chimique
2000
num. 7-8, p. 66-69.Asymmetric Synthesis of Actinoidic Acid Derivatives
Organic Letters
2000
Vol. 2 , num. 16, p. 2459-2462.DOI : 10.1021/ol006110s
A Novel Synthesis of Biaryl-Containing Macrocycles by a Domino Miyaura Arylboronate Formation: Intramolecular Suzuki Reaction
Organic Letters
2000
Vol. 2 , num. 22, p. 3477-3480.DOI : 10.1021/ol006520g
Inhibitory salt effect on the SNAr based macrocycloetherification of a linear diarylheptanoid
Synlett
2000
num. 3, p. 412-414.DOI : 10.1055/s-2000-6519
Synthesis of model of phomopsin-ustiloxin-type antimitotic agents
Synlett
2000
num. 9, p. 1363-1365.DOI : 10.1055/s-2000-7137
Synthesis of a model 22-membered AB-C-O-D ring of vancomycin containing biaryl and biaryl ether linkages
Tetrahedron Letters
2000
Vol. 41 , num. 11, p. 1747-1751.DOI : 10.1016/S0040-4039(00)00046-0
Recent progress in isolation, bioactivity evaluation and total synthesis of diarylheptanoids
Organic Preparations and Procedures International
2000
Vol. 32 , num. 6, p. 505-546.DOI : 10.1080/00304940009355948
1999
Total Synthesis of an Antitumor Agent RA-VII via an Efficient Preparation of Cycloisodityrosine
Journal of Organic Chemistry
1999
Vol. 64 , num. 17, p. 6283-6296.DOI : 10.1021/jo990432w
A high throughput synthesis of aryl triflate and aryl nonaflate promoted by a polymer supported base (PTBD)
Tetrahedron Letters
1999
Vol. 40 , num. 42, p. 7469-7472.DOI : 10.1016/S0040-4039(99)01529-4
A Unified Strategy toward the Synthesis of Acerogenin-Type Macrocycles: Total Syntheses of Acerogenins A, B, C, and L and Aceroside IV
Journal of Organic Chemistry
1999
Vol. 64 , num. 3, p. 914-924.DOI : 10.1021/jo981844s
An asymmetric total synthesis of sanjoinine G1
Tetrahedron Letters
1999
Vol. 40 , num. 1, p. 83-86.DOI : 10.1016/S0040-4039(98)80025-7
Design and synthesis of novel tridentate and tetradentate chiral ligands
Tetrahedron Letters
1999
Vol. 40 , num. 39, p. 7087-7090.DOI : 10.1016/S0040-4039(99)01454-9
4-Nitrophenyltriflate and 4-Nitrophenylnonaflate as New Perfluoroalkanesulfonyl Transfer Agents: Experimental and Computational Studies
Journal of Organic Chemistry
1999
Vol. 64 , num. 20, p. 7638-7642.DOI : 10.1021/jo990559l
Total synthesis and conformational studies of hapalosin, N-desmethylhapalosin and 8-deoxyhapalosin
Bioorganic & Medicinal Chemistry
1999
Vol. 7 , num. 5, p. 737-747.DOI : 10.1016/S0968-0896(98)00208-9
SNAr-based cycloetherification methodology: application in the synthesis of heterodectic macrocyclic peptides with endo aryl-aryl and aryl-alkyl ether bonds
Peptidomimetics Protocols; 1999. p. 293-320.ISBN : 0-89603-517-4
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Recent developments in reversing glycopeptide-resistant pathogens
Expert Opinion on Therapeutic Patents
1999
Vol. 9 , num. 8, p. 1005-1019.DOI : 10.1517/13543776.9.8.1005
1998
SNAr Based Cycloetherification Methodology: Application in the Synthesis of Heterodectic Macrocyclic Peptides with Endo Aryl-Aryl and Aryl-Alkyl ether Bonds
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Sciences Chimique
1998
Vol. 64 , p. 4-8.Synthesis of cycloisodityrosine revisited: A selective ring forming process
Tetrahedron Letters
1998
Vol. 39 , num. 7, p. 551-554.DOI : 10.1016/S0040-4039(97)10664-5
Chemoenzymic Synthesis of D-N-Boc-3,5- dihydroxy-4-methoxyphenylglycine
Journal of Organic Chemistry
1998
Vol. 63 , num. 16, p. 5662-5665.DOI : 10.1021/jo980233x
Horse liver esterase catalyzed enantioselective hydrolysis of N,O-diacetyl-2-amino-1-arylethanol
Tetrahedron: Asymmetry
1998
Vol. 9 , num. 1, p. 169-178.DOI : 10.1016/S0957-4166(97)00610-1
Approach towards the total synthesis of cyclopeptide alkaloids
Tetrahedron Letters
1998
Vol. 39 , num. 3/4, p. 283-286.DOI : 10.1016/S0040-4039(97)10513-5
Diastereoselective Synthesis of gamma -Hydroxy-beta -Amino Alcohols and (2S,3S)-beta -Hydroxyleucine from Chiral D-(N,N-Dibenzylamino)serine (TBDMS) Aldehyde
Journal of Organic Chemistry
1998
Vol. 63 , num. 5, p. 1709-1713.DOI : 10.1021/jo971468w
Asymmetric synthesis of 3,5-bis(isopropyloxy)-4-methoxyphenyl glycine by way of a diastereoselective Strecker reaction and an Evans electrophilic amination reaction
Tetrahedron: Asymmetry
1998
Vol. 9 , num. 17, p. 3095-3103.DOI : 10.1016/S0957-4166(98)00312-7
An efficient chloro-deamination procedure, application to the synthesis of advanced vancomycin C-O-D-O-E ring
Synlett
1998
num. 10, p. 1159-1161.DOI : 10.1055/s-1998-1857
A method for removal of N-Boc protecting groups from substrates on TFA-sensitive resins
Tetrahedron Letters
1998
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1997
Solution phase combinatorial synthesis of arylpiperazines
Tetrahedron Letters
1997
Vol. 38 , num. 23, p. 4091-4094.DOI : 10.1016/S0040-4039(97)00831-9
A formal total synthesis of deoxybouvardin
Tetrahedron
1997
Vol. 53 , num. 31, p. 10753-10764.DOI : 10.1016/S0040-4020(97)00706-0
Synthesis of model tricyclic C-O-D-O-E-F-O-G ring of teicoplanin
Tetrahedron Letters
1997
Vol. 38 , num. 33, p. 5795-5798.DOI : 10.1016/S0040-4039(97)01280-X
Novel vancomycin dimers with activity against vancomycin-resistant enterococci
Chemtracts
1997
Vol. 10 , num. 11, p. 818-821.Rapid and efficient solid phase syntheses of cyclic peptides with endocyclic biaryl ether bonds
Tetrahedron Letters
1997
Vol. 38 , num. 19, p. 3345-3348.DOI : 10.1016/S0040-4039(97)00654-0
First Total Synthesis of Acerogenin C and Aceroside IV
Journal of Organic Chemistry
1997
Vol. 62 , num. 22, p. 7544-7545.DOI : 10.1021/jo9714324
A highly stereoselective synthesis of (2S, 3S)-beta -hydroxyleucine
Tetrahedron Letters
1997
Vol. 38 , num. 10, p. 1771-1772.DOI : 10.1016/S0040-4039(97)00207-4
Synthesis of four atropdiastereoisomers of C-O-D-O-E ring of vancomycin by sequential cycloetherifications
Tetrahedron Letters
1997
Vol. 38 , num. 8, p. 1403-1406.DOI : 10.1016/S0040-4039(97)00036-1
Chemoenzymic synthesis of enantiomerically pure 4-fluoro-3-nitro and 3-fluoro-4-nitro phenylalanine
Tetrahedron: Asymmetry
1997
Vol. 8 , num. 3, p. 391-398.DOI : 10.1016/S0957-4166(96)00524-1
A novel strategy towards the total synthesis of cyclopeptide alkaloids. Reply
Angewandte Chemie, International Edition
1997
Vol. 36 , num. 10, p. 1074-1075.DOI : 10.1002/anie.199710742
4-Nitrophenyl triflate as a new triflating agent
Tetrahedron Letters
1997
Vol. 38 , num. 7, p. 1181-1182.DOI : 10.1016/S0040-4039(97)00024-5
SNAr-based macrocyclization via biaryl ether formation. Application in natural product synthesis
Synlett
1997
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1996
Synthesis of a model bicyclic C-O-D-O-E ring of vancomycin by a one-pot, double SNAr based macrocyclization
Chemical Communications
1996
num. 9, p. 1029-1030.DOI : 10.1039/cc9960001029
A New Approach to the Synthesis of Piperazinomycin and Bouvardin: Facile Access to Cycloisodityrosine via an Intramolecular SNAr Reaction
Journal of Organic Chemistry
1996
Vol. 61 , num. 2, p. 771-4.DOI : 10.1021/jo951375j
Synthesis of Modified Carboxyl Binding Pockets of Vancomycin and Teicoplanin
Journal of Organic Chemistry
1996
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Asymmetric Synthesis. 39.1 Synthesis of 2-(1-Aminoalkyl)piperidines via 2-Cyano-6-phenyl Oxazolopiperidine
Journal of Organic Chemistry
1996
Vol. 61 , num. 19, p. 6700-6705.DOI : 10.1021/jo960910s
Synthesis of hapalosin and 8-deoxy-hapalosin
Tetrahedron Letters
1996
Vol. 37 , num. 36, p. 6557-6560.DOI : 10.1016/0040-4039(96)01415-3
A novel strategy towards the total synthesis of cyclopeptide alkaloids
Angewandte Chemie, International Edition
1996
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Selective hydroxy group protection of gallic acid
Synthetic Communications
1996
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1995
Procédé de préparation de composés d’intérêt par cyclisation intramoléculaire et formation d’un pont éther biaryl
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- FR2716456 (B1)
- FR2716456 (A1)
- CA2183333 (A1)
- WO9522558 (A1)
1995
Palladium catalyzed reductive deprotection of alloc: Transprotection and peptide bond formation
Tetrahedron Letters
1995
Vol. 36 , num. 18, p. 3129-3132.DOI : 10.1016/0040-4039(95)00449-M
The first synthesis of a model bicyclic D-O-E-F-O-G ring of teicoplanin via sequential intramolecular SNAr reactions
Tetrahedron Letters
1995
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A new access to 14-membered macrocycle: synthesis of model F-O-G ring of teicoplanin
Tetrahedron Letters
1995
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Synthesis of a modified carboxylate-binding pocket of vancomycin
Tetrahedron Letters
1995
Vol. 36 , num. 27, p. 4781-4.DOI : 10.1016/0040-4039(95)00864-9
Asymmetric synthesis of (2S,3R) beta -(4-F-3-NO2) phenyl serine, D-(R)-4-methoxy-3,5-bistbutyldimethylsiloxy phenylglycine and their assemblage to C-O-D ring of vancomycin
Tetrahedron Letters
1995
Vol. 36 , num. 39, p. 7081-4.DOI : 10.1016/0040-4039(95)01409-B
A Convergent Synthesis of 14-Membered F-O-G Ring Analogs of the Teicoplanin Binding Pocket via Intramolecular SNAr Reaction
Journal of Organic Chemistry
1995
Vol. 60 , num. 20, p. 6389-96.DOI : 10.1021/jo00125a026
1994
A novel synthesis of K-13
Tetrahedron Letters
1994
Vol. 35 , num. 40, p. 7391-4.DOI : 10.1016/0040-4039(94)85322-3
An easy access to functionalized diaryl ethers: formal total synthesis of K-13
Tetrahedron Letters
1994
Vol. 35 , num. 31, p. 5649-52.DOI : 10.1016/S0040-4039(00)77270-4
SNAr-Based Macrocyclization: An Application to the Synthesis of Vancomycin Family Models
Journal of Organic Chemistry
1994
Vol. 59 , num. 19, p. 5535-42.DOI : 10.1021/jo00098a010
The first examples of SNAr-based macrocyclization: synthesis of model carboxylate-binding pockets of vancomycin
Journal of the Chemical Society, Chemical Communications
1994
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Reductive deprotection of aryl allyl ethers with Pd(Ph3)4/NaBH4
Tetrahedron Letters
1994
Vol. 35 , num. 25, p. 4349-50.DOI : 10.1016/S0040-4039(00)73351-X
1993
Elemental white phosphorus as a radical trap: a new and general route to phosphonic acids
Journal of the American Chemical Society
1993
Vol. 115 , num. 5, p. 2071-2.DOI : 10.1021/ja00058a082
A SNAr based facile synthesis of triaryl diethers, degradation products of vancomycin and related glycopeptide antibiotics
Tetrahedron Letters
1993
Vol. 34 , num. 48, p. 7741-4.DOI : 10.1016/S0040-4039(00)61553-8
Synthesis of various substituted dibenzo[b,d]pyranones including amino acid derivatives by SRN1 methodology
Heterocycles
1993
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A concise and efficient synthesis of protected actinoidic acid, the degradation product of vancomycin
Tetrahedron Letters
1993
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Asymmetric synthesis. 29. Preparation of 1,8-diazaspiro[5.5]undecane derivatives
Journal of Organic Chemistry
1993
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1992
An efficient procedure for the regioselective monoprotection of 1,2-diols
Tetrahedron
1992
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1991
Asymmetric synthesis. XXII. Formal synthesis of (-)-perhydrohistrionicotoxin
Tetrahedron Letters
1991
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1990
Study on the synthesis of some new biflavonoids. (VI). The catalytic hydrogenation of 3,3″-biflavones
Chinese Science Bulletin
1990
Vol. 35 , num. 9, p. 744-6.Synthesis of some new biflavonoids. IV. Synthesis of 3,3″-biflavone
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1990
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Synthesis of some new biflavonoids. (V). Total synthesis of O-hexamethyl brackenin
Gaodeng Xuexiao Huaxue Xuebao
1989
Vol. 10 , num. 6, p. 653-4.Synthesis of some new biflavonoids. I. Synthesis of the aromatic 1,4-diketones
Lanzhou Daxue Xuebao, Ziran Kexueban
1989
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Tetrahedron Letters
1989
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Asymmetric synthesis. XVIII. Preparation of chiral 1,2-diamines via the CN(R,S) method. Application to the synthesis of an analog of tetraponerine
Tetrahedron Letters
1989
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Synthesis of bisflavone-type compounds. (III). Selective demethoxylation of 1,4-bis(2′,4′,6′-trimethoxyphenyl)-1,4-butanedione
Lanzhou Daxue Xuebao, Ziran Kexueban
1989
Vol. 25 , num. 1, p. 157-8.Synthesis of some new biflavonoids. II. Synthesis of alpha ,alpha ‘-bichalcone
Huaxue Xuebao
1989
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Total synthesis of 3,3′-biflavone
Journal of the Chemical Society, Chemical Communications
1988
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